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(2S,4S)-4-(cyclooctylamino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
5-(3-methoxy-2,2-dimethylpropanoyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-6-methyl-4H-chromen-4-one
6-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
15-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-13-oxo-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
7-methoxy-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
1-methyl-4-(5-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)piperazine
N'1-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclopropane-1,1-dicarboxamide
1-(2-hydroxyethyl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
2-[3-(1H-imidazol-1-yl)pyrrolidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
3-ethoxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
1-[2-(4,4-difluoropiperidine-1-carbonyl)morpholin-4-yl]-2-(thiophen-3-yl)ethan-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[4-(furan-2-yl)phenyl]piperidin-4-amine
methyl 3-[(4-methoxyphenyl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(cyclohex-3-en-1-ylmethyl)-4-(4-methoxyphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
ethyl 3-benzyl-1-(1-propylpiperidin-4-yl)piperidine-3-carboxylate
4-methoxy-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}pyrimidin-2-amine
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
5-cyclopropyl-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(methylsulfamoyl)ethyl]benzamide
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
2-butyl-8-(2,3-difluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
4-chloro-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1-methyl-1H-indazole
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-N-phenylpropanamide
methyl 1-[(3S,5S)-1-[(2-chlorophenyl)methyl]-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(3-chloro-4-methoxyphenyl)-6-[2-(4-methylphenoxy)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aS,8aR)-6-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N,1,4,6-tetramethyl-2-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-yl)ethan-1-one
2-benzyl-4-(pyrrolidine-1-sulfonyl)morpholine
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
5-(2,6-dimethoxyphenyl)-N-(pyridin-3-yl)furan-2-carboxamide
6-methyl-2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-{2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(propan-2-yl)-4-[3-(pyridin-4-yl)propanoyl]-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(1R,3R)-N1-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]cyclopentane-1,3-diamine
N-[2-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
6-fluoro-N-[2-(2-methylpropanesulfonyl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-methyl-5-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]-N-(thiophen-2-ylmethyl)-1,3-thiazol-2-amine
2-(morpholin-4-yl)-N-(2-phenoxyethyl)-2-(pyridin-3-yl)acetamide
3-[3-({[2-(2,6-dimethylphenoxy)ethyl](methyl)carbamoyl}amino)phenyl]-N-methylpropanamide
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
1-(azepan-1-yl)-3-(4H-1,2,4-triazol-4-yl)propan-2-ol
(3R,7S,8aS)-3-benzyl-7-{[(2-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione