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2-chloro-6-methoxy-4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenol
1-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]but-3-en-1-one
1-{4-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}imidazolidin-2-one
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
2-[(4-methoxyphenyl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
{5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
4-methyl-3-[(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)sulfanyl]-4H-1,2,4-triazole
5-fluoro-N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(oxolan-2-ylmethyl)benzamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[3-(morpholin-4-yl)propyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
methyl 2-chloro-4-{[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]amino}benzoate
(3R,4R)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
9-methoxy-N-methyl-3-[2-(methylsulfanyl)benzoyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(pyrrolidin-1-yl)propyl]amine
N-[(3R,4S)-1-(5-chloro-2-methylpyrimidine-4-carbonyl)-4-cyclopropylpyrrolidin-3-yl]methanesulfonamide
4-{3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperazin-2-one
N-(2,5-dimethyl-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrrol-1-yl)acetamide
1-{1-[(4-cyanophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]hept-6-ynamide
(1S,3R)-3-amino-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)cyclopentane-1-carboxamide
2-{5-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(2-oxoazonan-1-yl)acetamide
N-methyl-6-oxo-1-(3-phenylpropyl)-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-[6-(2,4,6-trimethylphenyl)pyridazin-3-yl]thiomorpholine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
4-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-1,4-oxazepan-6-ol
2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
1-(3-methoxybenzoyl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-(3-methoxyphenyl)-1,2,4-triazine
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(3S,4S)-4-methoxypyrrolidin-3-yl]-2,6,8-trimethylquinoline-4-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
3-{3-cyclohexyl-1-[4-(2-hydroxyethyl)piperazin-1-yl]prop-2-yn-1-yl}benzonitrile
2-(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(propan-2-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2-oxazole-5-carboxamide
1-[3-(3-fluorophenyl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(3S,4R)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
[1-({4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-3-yl]methanol
4-methoxy-N-(2-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
(3aR,6aS)-1-oxo-5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenol
1-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
(2S,4R)-4-amino-N-(propan-2-yl)-1-(pyridine-2-carbonyl)pyrrolidine-2-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylprop-2-ynamide