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6-ethyl-4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-2-methylquinoline
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}propanamide
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-(3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidin-1-yl)acetamide
8-cyclohexyl-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(2-methylphenyl)methyl]benzamide
5-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]amine
3-(1,2-oxazinan-2-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
N-[3-(furan-2-yl)propyl]-2-(1H-pyrazol-1-yl)benzamide
4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]-N-propylpiperidine-1-carboxamide
2-{4-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1-cycloheptyl-N-methyl-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-5-methyl-1H-pyrrol-1-yl)pyridine
4-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-3-yl}pyrimidine
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
2-({4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
1-(5-amino-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
4-(2-methyl-1H-imidazol-1-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-oxo-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,2-dihydroquinoline-4-carboxamide
8-cyclopropanecarbonyl-2-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-(2-chloro-4-fluorophenyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1H-imidazol-1-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)butan-1-one
N-({3-methyl-7-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
1-{[2-(2-aminoethyl)quinazolin-4-yl]amino}-3-(3-methoxyphenoxy)propan-2-ol
N-{4-[5-methyl-4-({2-[3-(trifluoromethyl)phenyl]acetamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide
4-{[4-(naphthalen-2-yl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N,1-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-(4-fluorophenyl)-4-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]butane-1,4-dione
6-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N,N-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-(2-ethylphenyl)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
N,N-dimethyl-5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
methyl 3-acetamido-1-ethyl-5-[(1,2,3,4-tetrahydronaphthalen-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(5S)-5-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
6,7-dimethyl-2-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}-1H-1,3-benzodiazole
(1S,6R)-3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(pyridin-3-yl)-5-[4-(thian-4-yl)piperazine-1-carbonyl]pyrimidine
5-{1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(2-methoxybenzoyl)-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
5-methyl-1'-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(thiomorpholin-4-yl)-3-{2-[({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-phenylpyrimidine-5-carboxamide
4-(4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
6-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
1-(propan-2-yl)-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
8-[(8-fluoroquinolin-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(6-methylpyridin-2-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine