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2-(1H-indazol-1-yl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-amino-6-(3-hydroxyphenyl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-(4-fluorophenyl)-4-(2-methoxypyridine-4-carbonyl)-1,4-diazepane
N-[2-(furan-2-yl)ethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
2,2-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}butanamide
(3aR,6aR)-2-(2-hydroxyethyl)-5-[3-(3-methoxyphenyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2,5-difluoro-4-(trifluoromethyl)phenyl]-1-[3-(3-oxopiperazin-1-yl)propyl]urea
3-(2,5-difluorobenzoyl)-1-[(2-ethoxyphenyl)methyl]piperidine
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
2-(morpholin-3-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
(2R,3R,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 9-(cyclopentyloxy)-7-oxo-3-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxo-N-(propan-2-yl)acetamide
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-ethoxyethan-1-one
2-{4-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}-4-methyl-6-(propan-2-yl)quinazoline
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3-(propan-2-yl)-1,2-oxazole
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
4-[1-(4-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)ethyl]morpholine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(3-{3-[4-(5-amino-3-methyl-1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-5-yl}piperidin-1-yl)ethan-1-one
(3R,4R)-3-cyclobutyl-4-methyl-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-ol
5-acetyl-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]thiophene-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-(pentan-3-yl)-N-(2-phenylethyl)propanamide
N-[(2S)-1-oxo-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-2-yl]acetamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 1-[1-(methylsulfanyl)propan-2-yl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-[(2-chlorophenyl)methyl]-N-[(5-fluoro-2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-acetamido-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazole-7-carboxamide
N-{4-chloro-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}acetamide
(3R,4R)-1-(5-chloro-2-methylpyrimidine-4-carbonyl)-4-ethylpiperidine-3,4-diol
(2R,6S)-2,6-dimethyl-4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)morpholine
2-[hydroxy(phenyl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
5-fluoro-2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-(pyrrolidin-1-yl)pyrimidine
(2S,4S)-4-amino-N-methyl-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-[2-(pyridin-2-yl)ethyl]acetamide
N-cyclobutyl-3-[(oxan-2-ylmethyl)sulfamoyl]benzamide
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-(azepan-1-yl)-3-{4-chloro-2-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
5-ethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
2-[1-methyl-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl]ethan-1-ol
4-[(2-methylpyridin-3-yl)oxy]-1-[2-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
(4aR,7aS)-1-acetyl-4-[3-(4-methoxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-fluoro-2-methyl-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]quinoline
5-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1,7-dimethyl-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
N-cyclopentyl-N'-ethyl-N'-[(2E)-3-phenylprop-2-en-1-yl]butanediamide