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{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
2-{1-cyclopentyl-4-[(8-methoxyquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-fluoro-4-methoxyphenyl)-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
N-[4-methyl-3-({[3-(1H-1,2,3-triazol-1-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
4-phenyl-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine-4-carboxylic acid
(2S)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2-phenylethan-1-ol
3,5-dimethyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-pyrrole-2-carboxamide
N-({7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]propanamide
N-cyclohexyl-N-ethyl-2-(4-fluorophenoxymethyl)-4-hydroxypyrimidine-5-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-N'-(2-chlorophenyl)ethanediamide
1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(quinolin-5-ylmethyl)amine
N-[2-(3-hydroxyphenyl)pyridin-3-yl]cyclopropanecarboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(2,5-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(benzyloxy)-8-(3-phenylprop-2-ynoyl)-1,8-diazaspiro[4.5]decan-2-one
6-(4-chlorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
methyl 6-[2-(2-fluorophenyl)acetyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-({2-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-ethyl-2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
2-(4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
(5S,9aS,9bS)-2-cyclopentyl-5-(3,4-dimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[4-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethoxy)phenyl]propanamide
2-(2-fluoro-6-hydroxybenzoyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methoxypyrimidine-5-carboxamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-2-phenylpiperazine
4-[2-(2-ethoxyphenoxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
N4-methyl-N4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-6-(propan-2-yloxy)pyrimidine-2,4-diamine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(4-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
N-(1-benzyl-1H-pyrazol-5-yl)-2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
N-(4-{4-[(3-ethoxypropyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
ethyl 5-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-(furan-3-ylmethyl)-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-methylazepane-2-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-phenylpyridazin-3-amine
6-methoxy-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-[(4-fluorophenyl)methyl]piperidin-3-yl)methanol
2-(4-fluorophenyl)-1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
1-[2-(adamantan-1-ylformamido)ethyl]-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
4-(dimethylamino)-N,N-bis(propan-2-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-butyl-N-[2-(diethylamino)ethyl]-N-ethyl-1,3-benzoxazole-5-carboxamide
3-(2,4-difluorophenyl)-1-[2-(dimethylamino)ethyl]-6-(4-hydroxybutan-2-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one