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2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
2-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5,5-dimethyl-3-(2-oxo-2-{4-oxo-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-1'-yl}ethyl)-1,3-oxazolidine-2,4-dione
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-[2-(dimethylamino)ethyl]-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
2-oxo-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
9-(3-phenylpropyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
(5S,9aS,9bS)-5-(2,3-dimethoxyphenyl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[(3R,4R)-1-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-(2-{[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}propyl)-3,4-dihydroquinazolin-4-one
methyl 2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(9H-fluoren-2-yl)-1-(pyrrolidin-3-yl)-1H-imidazole
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
N6-cyclopropyl-N5-(isoquinolin-5-ylmethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-methyl-N-[3-(4-methylpiperazine-1-carbonyl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[3-(morpholin-4-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(2,3,6-trimethylphenoxy)acetamide
6-(methoxymethyl)-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4S)-4-[4-(2-fluoro-5-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
4-[(4,6-dimethylpyrimidin-2-yl)amino]-1-methylpyrrolidin-2-one
N-(2-methylpropyl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}-N-(thiophen-3-ylmethyl)acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-oxo-2-phenyl-N-(pyridin-3-ylmethyl)acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(4-{[1-(thiophen-2-ylmethyl)piperidin-3-yl]amino}quinazolin-2-yl)methanol
N-(2-methoxyethyl)-N-methyl-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-methyl-3-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-2-(morpholin-4-yl)quinoline
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbut-2-en-1-yl)piperidine
2-(3-methoxypropyl)-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-3-methoxy-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)propanamide
N-{[7-(2,4-dimethylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
5,6-dimethyl-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazole
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[3-(azepan-1-ylmethyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
8-fluoro-2-({4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
1-cyclopentyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-4-carboxamide
(2R,6S)-4-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,6-dimethylmorpholine
6-ethyl-3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,5-dimethyl-1,2-dihydropyridin-2-one
1-cyclopropyl-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
dimethyl({[5-(2,3,4,9-tetrahydro-1H-carbazol-7-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-4-propylpyrimidine-5-carboxamide
1-[3-(furan-2-yl)propanoyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-amine
{1-[6-(4-fluorophenyl)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]pyridin-2-yl]piperidin-3-yl}methanol
2-(pyrrolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}benzamide
N-methyl-5-(oxolan-2-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
4-ethyl-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
3,5-dimethyl-4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-oxazole