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6-[2-(benzyloxy)phenyl]pyrazine-2-carboxylic acid
13-(5-tert-butyl-1H-pyrazol-3-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(oxolan-2-ylmethyl)piperazin-1-yl]ethan-1-one
[(3-tert-butyl-1H-pyrazol-5-yl)methyl][(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
(3S)-4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,3-dimethylpiperazin-2-one
1-[4-(6-hydroxy-1,4-oxazepane-4-carbonyl)phenyl]imidazolidine-2,4-dione
N-(1-benzylpiperidin-3-yl)-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-4-methyl-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-5-carboxamide
N-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
(4aS,8aR)-1-(3-aminopropyl)-6-(ethanesulfonyl)-decahydro-1,6-naphthyridin-2-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]butanamide
2-butoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-(4-fluorophenyl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
2-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-1-methyl-1H-1,3-benzodiazole
methyl 1-[3-(cyclopropylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-phenylpropyl)propanamide
7-methyl-3-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1,7-dimethyl-1H-indole-2-carboxamide
2-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-N-(2-fluoro-4-methylphenyl)acetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-hydroxy-2-(pyridin-4-yl)pyrimidine-5-carboxamide
(1R,3S)-3-ethoxy-7-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
N-{[5-(4H-1,2,4-triazol-3-ylsulfanyl)furan-2-yl]methyl}pyridin-3-amine
(4aR,6R,8aS)-2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
5-fluoro-3-methyl-2-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1H-indole
2-(4-fluorophenoxymethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
(4aS,7aR)-1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
dimethyl({2-[4-(2-methyl-1-benzofuran-7-carbonyl)morpholin-2-yl]ethyl})amine
4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-thiazole
propan-2-yl 2-chloro-5-[2-(1H-1,2,4-triazol-1-yl)propanamido]benzoate
8-(2,3-dihydroxybenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-3-cyclopentyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
1-(naphthalen-1-ylmethyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
methyl 8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2,3-dimethoxy-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
4-[7-(1-ethyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
2-methyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]-4-phenylpiperidin-4-ol
2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(methylsulfamoyl)ethyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
methyl 3-[2-(3,5-difluorophenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]morpholine-4-sulfonamide
N3-methyl-1-(3-methylbutyl)-N5-[(3-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide