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N-[2-(2-chlorophenyl)ethyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
1-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
6-(methoxymethyl)-1-methyl-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 5-(1-benzoylpiperidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]pyrimidin-2-yl}benzenesulfonamide
(1S,4S)-5-(1-benzothiophen-2-ylmethyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{5-[2-(propan-2-yl)pyrimidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,2-oxazol-3-ylmethyl)propanamide
4-(1H-1,3-benzodiazol-1-yl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
N-[1-(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
7-(5-propyl-1,2-oxazole-3-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(5-methylthiophen-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
4-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methyl-1,3-thiazol-2-amine
6-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
N-(3,4-dichlorophenyl)-4-(dimethylamino)azepane-1-carboxamide
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}piperidin-4-ol
methyl 2-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}butanoate
1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
5-{3-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
3-[(1-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propan-2-yl)oxy]pyridine
1-(diethylamino)-3-{5-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
3-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-N,N-dimethylpiperidine-1-carboxamide
3-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)-1-methylpyrrolidine-2,5-dione
methyl 1-(2-methylpropyl)-5-[(3-phenylpropyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
N-[(3S,4R)-1-(4-aminopyrimidin-2-yl)-4-propylpyrrolidin-3-yl]acetamide
(2S,4S)-4-amino-1-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
[2-(2-ethylphenoxy)ethyl](furan-3-ylmethyl)amine
2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
1-{3-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzoyl}piperidine
1-(1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-phenylpropan-1-one
5-(1-cyclopentyl-1H-pyrazol-3-yl)-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,3-thiazol-2-amine
1-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-1H-1,2,4-triazole
3-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-N-phenylpropanamide
N-(2-methylpropyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-[2-(4-methoxyphenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-(4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-1H-1,3-benzodiazole
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
[(5-{1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]dimethylamine
N-methyl-N'-(4-methylphenyl)-N-(oxan-2-ylmethyl)propanediamide
4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-2-(prop-2-en-1-yl)phenol
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-(4-fluorophenyl)-2-oxo-2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione