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N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
7-(3-methoxyphenyl)-2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4,6-dimethyl-3-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-{3-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
ethyl 2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetate
4-[(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-2-yl)methyl]morpholine
5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
1-(4-methanesulfonylpiperazin-1-yl)-3-(pyridin-4-yl)propan-1-one
N-cycloheptyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-{5-[(6-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
N-[(3R,4S)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]propane-1-sulfonamide
N2,N2,5,6-tetramethyl-N4-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-2,4-diamine
(1R,2R,4R)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-2-(2-methylphenyl)acetamide
N-cyclopropyl-4-methyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
(5S,9aS,9bS)-5-(2-fluoro-4-methoxyphenyl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-methoxy-3-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1-benzofuran-2-carboxamide
3-(1H-pyrazol-1-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]benzamide
N-[2-(4-chlorophenyl)ethyl]-N-(pyridin-4-ylmethyl)oxane-2-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]cyclohexanecarboxamide
2-(5-tert-butyl-1H-pyrazol-3-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine-3-carboxamide
2-(3,4-dimethoxyphenyl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)quinolin-4-ol
2-({2-[bis(prop-2-en-1-yl)carbamoyl]phenyl}amino)acetic acid
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)acetamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
2-methyl-5-{3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]phenyl}-1,3,4-thiadiazole
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2S)-1-(piperidin-4-yl)pyrrolidine-2-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
[(1-benzylpiperidin-4-yl)methyl](methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-phenyl-4-[1-(2,3,4-trimethoxybenzoyl)piperidin-3-yl]piperazine
8-(4-methyl-1H-imidazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,4-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(2-fluorophenyl)-N-[(1S,2R)-2-{[1-(4-methylphenyl)piperidin-4-yl]amino}cyclobutyl]acetamide
N-[3-(cyclopentyloxy)propyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-[2-(2-methoxyphenoxy)ethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-3-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[2,1-b][1,3]thiazol-6-ylmethyl})amine
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl]acetamide
1-[4-(2-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-8-methylquinazolin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-(2-methoxyphenyl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
2-methyl-5-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2,3-dihydro-1H-isoindole-1,3-dione
7-[(4-chlorophenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(1-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide