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2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
[1-({[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]amino}methyl)cyclopentyl]methanol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)isoquinoline-5-carboxamide
2-phenyl-N-[3-(pyridin-3-yloxy)propyl]imidazo[1,2-a]pyridine-6-carboxamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
1-methyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(2-methylphenyl)benzamide
2-(4-methoxyphenoxymethyl)-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,3-oxazole
N-[3-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)-2-methylphenyl]furan-2-carboxamide
3-[(2,3-dimethoxyphenyl)methyl]-5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
2-(5-fluoro-4-methoxypyrimidin-2-yl)-N,N-bis(propan-2-yl)benzamide
2-ethyl-9-[(2,3,4-trifluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-2-ylmethyl}-3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazole
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(propan-2-yloxy)acetamide
methyl 2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}piperidine-1-carboxylate
(3aS,7aR)-5-methyl-2-(1-phenylcyclopentanecarbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
6-(4-chlorophenyl)-N-[1-(pyridin-2-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4R)-4-amino-1-[4-methoxy-3-(methoxymethyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
N-ethyl-2-(1-methyl-1H-pyrrol-3-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
3-amino-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
N-(furan-2-ylmethyl)-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
N-cyclopentyl-4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)benzamide
methyl 2-(azocane-1-sulfonyl)-6-(4-methyl-2-oxopentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2-[3-(trifluoromethoxy)phenyl]pyrimidin-4-yl}piperidin-3-ol
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
N,N-dimethyl-5-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
(2E)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-phenylprop-2-en-1-one
1-[3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenyl]imidazolidin-2-one
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
2-[1-(2H-1,3-benzodioxol-5-yl)-5-methyl-1H-1,2,4-triazol-3-yl]acetamide
1-{4-[3-(morpholin-4-ylmethyl)phenyl]phenyl}cyclopentane-1-carbonitrile
N-[2-(3-methoxyphenyl)-1-[1-(2-methylbenzoyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-(2,3-dihydro-1H-inden-4-yl)-5-[2-(methylsulfanyl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
{4-benzyl-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-4-yl}methanol
(1R,5R)-6-(5-ethyl-1,3-oxazole-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
6-ethyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-2-methyl-1H-imidazole
methyl (2S)-1-{7-acetamido-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazole-5-carbonyl}pyrrolidine-2-carboxylate
3-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
2-benzyl-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,3-benzoxazole-5-carboxamide
(3aR,6aR)-2-[2-(3-methoxyphenyl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
6-methyl-2-({2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
5-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[(2-fluorophenyl)methyl]-3-(2-methylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
7-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide