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2-{2-[1-(4-phenyl-1,3-thiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4-hydroxy-N-[1-(4-methanesulfonylphenyl)propyl]-2-methylpyrimidine-5-carboxamide
4-{4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1-(2-methoxyethyl)pyrrolidin-2-one
3-(3-methoxyphenyl)-N-(2-oxoazepan-3-yl)-1H-pyrazole-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
1-(cyclopent-1-ene-1-carbonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
4-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}phenol
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-phenylacetamide
N-{[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
2-(5-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-[4-(ethanesulfonyl)piperazin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
2-(2-methylpropyl)-8-[(3-methylquinoxalin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
4-methyl-2-[1-(3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-4-ylmethyl)amine
3-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyridine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbenzamide
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(4-fluorophenoxy)piperidine
N-[3-(1H-indol-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxamide
{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-ethyl-N-(2-methoxyethyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-6-methyl-3-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 3-[(2-fluorophenyl)methyl]-1-(3-methoxypropanoyl)piperidine-3-carboxylate
N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
4-ethyl-2-methyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(piperazin-1-yl)propan-1-one
N-[(4-methoxypyridin-2-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
methyl 5-(cyclopentylamino)-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-[1-(1H-indol-5-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
(3S)-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,3-dimethylpiperazin-2-one
N-ethyl-2,5-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
8-(cyclohexylmethyl)-3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
3-(3-methoxyphenyl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-5-carboxamide
N-{4-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenyl}acetamide
2-(1H-imidazol-1-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]acetamide
7-(cyclopropylmethyl)-2-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-fluoropyridine
N-ethyl-2-[4-(6-methoxy-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperazin-1-yl]acetamide
2-(2-hydroxyethyl)-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3,4-trimethoxybenzamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(2-methylfuran-3-carbonyl)piperidine-4-carboxylic acid
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-methoxyphenoxy)acetamide