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6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-(propan-2-yl)pyrimidin-4-amine
2-{4-[1-(2-methoxyphenyl)piperidin-4-yl]-1-methylpiperazin-2-yl}ethan-1-ol
2-[2-(3-fluorophenyl)ethyl]-4-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
5-({2-[(4-methylpyridin-2-yl)amino]ethyl}carbamoyl)-2,1,3-benzoxadiazol-1-ium-1-olate
2-{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-1-yl}-1,3-benzoxazole
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
7-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 3-(2,6-difluorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{5-[(5-fluoro-2-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
N-[(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
3-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-5-methoxyphenol
2-[3-(4-methanesulfonylphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
(dicyclopropylmethyl)(methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
3,3-dimethyl-1-[(3S,4R)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-ethyl-2-(2-methoxy-5-methylphenyl)pyrimidine
{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
methyl 1-ethyl-5-{[(4-methylphenyl)methyl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
N-(3,3-diphenylpropyl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
4-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-3-fluoropyridine
1-(4-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}phenyl)ethan-1-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
N-[2-(azepan-1-yl)ethyl]-1-(2-hydroxyethyl)-N-(propan-2-yl)piperidine-3-carboxamide
2-ethyl-6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-(1-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
(4aS,7aR)-1-(2-chlorobenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,9aR)-1-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-octahydro-1H-quinolizin-1-ol
1-{2-[4-(3-phenylpropyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(methylsulfanyl)pyrimidine-5-carboxamide
N-{4-[1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-imidazol-2-yl]phenyl}acetamide
4-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2-phenylmorpholine
6-(2H-1,3-benzodioxol-5-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-N,N-diethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-(5-{12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}furan-2-yl)benzonitrile
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl][(8-methoxy-2H-chromen-3-yl)methyl]methylamine
1-({4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]phenyl}methyl)azepane
1-ethyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{2-[5-(3,3-dimethylpyrrolidine-1-carbonyl)thiophen-2-yl]pyrrolidine-1-carbonyl}-1-methyl-1H-pyrrole
5-(3,5-dimethylphenyl)thiophene-2-carboxamide
1-ethyl-5-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]piperidin-2-one
3-[4-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-N-(pyridin-2-ylmethyl)aniline
2-[1-(pyridine-3-sulfonyl)pyrrolidin-3-yl]benzoic acid