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3-[1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2-{9-[(3-chloro-4-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
(1S,5R)-3-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3,9-diazabicyclo[3.3.2]decan-10-one
3-[(3R,4S)-1-(4-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(3-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}phenoxy)acetamide
7-methyl-2-(1H-pyrazol-4-yl)-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]quinoline
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methylphenoxy)piperidine
2-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}piperazin-1-yl)pyrimidine
2-(1-ethylpiperidin-4-yl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}ethan-1-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
5-oxo-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
(3S,9aR)-3-(2-methylpropyl)-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
{[(1R,5S,6S)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
5-acetyl-N,2,4-trimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrrole-3-carboxamide
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidine-3-carbonitrile
(2E)-3-(2-chlorophenyl)-1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)prop-2-en-1-one
methyl[(5-methylfuran-2-yl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
9-(4-chloro-2-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
(4aR,7aS)-1-benzyl-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-methylphenyl)methyl]-4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperazin-2-one
(1H-1,3-benzodiazol-2-ylmethyl)[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
[5-(1H-imidazol-1-yl)-2-methoxyphenyl]methanol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-2-yl)-4-(trifluoromethyl)pyrimidine-5-carboxamide
4-(2-ethylpyrimidin-4-yl)-5,6,7-trimethoxy-1,2,3,4-tetrahydroquinolin-2-one
3-methyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
3-methyl-5-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
ethyl 2-({[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]carbamoyl}amino)acetate
ethyl 4-[4-(4-{[2-(piperidin-1-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
4-methoxy-2-({3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-cyclopropyl-3-methyl-1H-pyrazole-4-carboxamide
N-(4-sulfamoylphenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
3-(furan-2-ylmethyl)-5-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1'-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N2-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-N4,N4-dimethylpyrimidine-2,4-diamine
3-{[1-(3-methanesulfonamidopropanoyl)piperidin-4-yl]methyl}benzoic acid
2-[(3,5-difluorophenyl)methyl]-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
5-butyl-1'-[(2,2-dimethyloxan-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(pyridin-3-yl)propan-1-one