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4-{[2-(4-methoxyphenoxy)phenyl]methyl}morpholine
N6-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[1-(3-cyclopentylpropyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[(5-propyl-1H-pyrazol-3-yl)methyl]amine
[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
1-(1,3-benzoxazol-2-yl)-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-amine
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methylpropanamide
9-[2-(1H-imidazol-1-yl)propanoyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
4,6-dimethyl-2-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
N-cyclopropyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-(thiophen-3-ylmethyl)propanamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(diphenylmethyl)piperazine
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(1-propylpiperidin-4-yl)acetamide
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
N-(3-cyclopentylpropyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-(1-ethylpiperidin-4-yl)-N-methyl-2-(pyrazin-2-yl)acetamide
4-[(2S)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carbonyl]morpholine
7-(2,1,3-benzoxadiazol-4-ylmethyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(propan-2-yl)pyridin-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
methyl 3-(cyclohex-3-ene-1-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(cyclohexylmethyl)-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
2-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amine
1-benzyl-5-[(furan-2-ylmethyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{2-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
N-butyl-2-[methyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]acetamide
2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
1,3-dimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-{2-[5-(6-methylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
N-[(1-cyclohexylpiperidin-3-yl)methyl]-4-phenyl-N-(pyridin-3-ylmethyl)butanamide
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-[(2-methyl-1,3-thiazol-4-yl)methyl]urea
2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-6-methoxyphenol
2-(4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
2-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-butyl-4-(4-hydroxyquinoline-2-carbonyl)-1-methylpiperazin-2-one
4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[6-(dimethylamino)pyrimidin-4-yl]pyrrolidine-3-carboxylic acid
N-[(3S,4R)-1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
1-{2-[4-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-5-methylpyrrolidin-2-one
ethyl 2-[1-(hydroxymethyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetate
2-(5-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}furan-2-yl)benzonitrile
2-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
5-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
3-methyl-7-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one