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N-(1-methyl-1H-indazol-3-yl)-2-[2-(4-methylbenzoyl)-1H-imidazol-1-yl]acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-2-(1H-pyrazol-1-yl)benzamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-(2-aminoethyl)-N-[2-(quinolin-8-yloxy)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
methyl 4-(4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)benzoate
8-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
3-[2-(2,4-difluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine
4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-(2-methoxyethyl)-4-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}morpholine
(4aS,7aR)-N-(2-ethylphenyl)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-cyclopropyl-9-[(2,3-difluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[3-oxo-3-(3-oxo-4-phenylpiperazin-1-yl)propyl]methanesulfonamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(4-methoxyphenyl)-2-methylpiperazine
(3S,4S)-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-(3-methoxybenzoyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
7-(3-chlorophenyl)-4-[2-(morpholin-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,8-dimethylquinoline-4-carboxamide
2-(4-cyclopentylpiperazin-1-yl)-2-(3-hydroxyphenyl)acetic acid
2-ethyl-N-(furan-2-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}butanamide
(7S,9aR)-7-[(2S)-butan-2-yl]-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
5-methoxy-9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1-oxa-9-azaspiro[5.5]undecane
4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)morpholine
7-(1-benzothiophen-3-yl)-4-(furan-2-ylmethyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(but-2-yn-1-yl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(furan-2-ylmethyl)amine
(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-[(2R,3R)-2-methoxy-1'-(4-methyl-2-oxopentanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-2-propyl-1,3-thiazole
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(thiophen-2-ylmethyl)propanamide
3-(2H-1,3-benzodioxol-5-yl)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)propan-1-one
3-(1,3-dimethyl-1H-pyrazol-5-yl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6,6-dimethyl-1-(4-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-({[(2-methyl-1-benzothiophen-3-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetic acid
N3-methyl-4-oxo-1-(2-phenylethyl)-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
5-[({1-[3-(4-chlorophenyl)phenyl]piperidin-4-yl}amino)methyl]pyrrolidin-2-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
2-{5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-(3-hydroxy-3-methylbutyl)-N-[(1-hydroxycyclohexyl)methyl]benzamide
5-(1H-imidazol-1-ylmethyl)-2-(6-methoxypyridin-3-yl)pyridine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(morpholin-4-yl)pyridine-3-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)cyclohexanecarboxamide
2-(3-acetyl-1H-indol-1-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one