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2-[2-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-1H-indole-6-carboxamide
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
(4S)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
5-cyano-6-(2,3-dimethoxyphenyl)-2-methylpyridine-3-carboxylic acid
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](quinolin-4-ylmethyl)amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
N-{[7-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-{[5-(3-methylpyrazin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[4-({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}amino)-6-methylpyrimidin-2-yl]phenol
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
9-(2-aminopyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(hydroxymethyl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-cyclopropyl-4-phenyl-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(2-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N,N-dimethyl-5-[4-(2-methylpiperidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
4-methyl-6-{3-[(methylsulfanyl)methyl]piperidin-1-yl}-5-(prop-2-en-1-yl)pyrimidin-2-amine
(1S,5R)-6-(2-chloro-4-fluorobenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyrazine-2-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
3-[5-chloro-2-(propan-2-yloxy)phenyl]-12-methyl-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
2-benzyl-N-[(1S)-1-(4-chlorophenyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-cyclohexyl-N-(oxan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-(1-benzofuran-2-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3,4-dichlorophenyl)-N-ethyl-N-methylmorpholine-4-sulfonamide
1-methyl-3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
4-[6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
N-(furan-2-ylmethyl)-2-{3-[3-(3-methylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(3-methoxyphenyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
ethyl 3-(2-phenylethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
ethyl 2-({[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)amino)acetate
2,3-dimethoxy-N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)benzamide
1-cyclohexyl-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-4-carboxamide
4-oxo-4-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}butanamide
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-4-(piperidin-1-yl)butan-1-one
4-{[3-(1H-indol-1-yl)propyl]amino}-1λ4-thian-1-one
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(5-methyl-1,3-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]-N,N-dimethylpiperidine-1-carboxamide
6-(2-chloro-4-fluorobenzoyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(2R,4R,6S)-2-tert-butyl-6-(1,5-dimethyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-(thiophen-2-yl)azetidine