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8-[6-hydroxy-2-(propan-2-yl)pyrimidin-4-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
ethyl 2-{3-[3-(pyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}acetate
(5-{1-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-(pyridin-3-yl)propan-1-one
1-(2-methoxy-5-{[methyl(2-phenylethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
3-(1H-indol-3-yl)-1-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
4-(hydroxymethyl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-ol
methyl 3-(3-cyclopentylpropanoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1,3-benzothiazol-2-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
2-[3-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)phenoxy]acetamide
3-cyclohexyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)pyrrolidine-1-carboxamide
N-[(2S,4R,6S)-2-ethyl-6-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]oxan-4-yl]benzamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-(2-methylpropyl)-4-[3-(2-oxopyrrolidin-1-yl)benzoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(1-propylpiperidin-4-yl)benzamide
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl})[1-(pyrazin-2-yl)propan-2-yl]amine
5-cyclopropanecarbonyl-1'-(6-ethyl-2-methylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,8aR)-6-(pyridin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-butyl-1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-(3-hydroxy-3-methylbutyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]benzamide
(1R,5S,8S)-3-{[2-(benzylamino)pyrimidin-5-yl]methyl}-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
(1R,3S)-3-ethoxy-7-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
4-[(2S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
4-chloro-5-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
(1S,6R)-9-[(2-phenylphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(4-fluorophenyl)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)-N-methylpiperidine-3-carboxamide
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N,N-dimethyl-5-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}-1,3-thiazol-2-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
7-(1-benzothiophen-3-yl)-4-[(5-methylfuran-2-yl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxobutanamide
5-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-[5-(2-methyl-1-benzofuran-7-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(3S,9R)-11-(4-chlorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[2-(4-fluorophenyl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]pyrimidin-4-yl}piperidin-3-ol
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(methylsulfanyl)propyl]acetamide
methyl 1-oxo-2-(1,3-thiazol-4-ylmethyl)-1,2-dihydroisoquinoline-7-carboxylate
7-(cyclohexylmethyl)-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-5-{1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-ethyl-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-N-(thiophen-2-ylmethyl)acetamide
5-(6-hydroxy-1,4-oxazepane-4-carbonyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]pyrrolidine-1-carboxamide