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2-methyl-5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
N2-[2-(cyclohexylsulfanyl)ethyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
N-(3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)acetamide
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
8-(6-aminopyridine-3-carbonyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-benzylpiperidin-3-yl)-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}-N-[2-(propan-2-yloxy)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N,N-dimethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrazine-2-carboxamide
(benzylsulfamoyl)({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
7-(pyridin-3-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(2-methylphenyl)methyl]-3-(oxan-4-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-(1-methyl-1H-imidazol-2-yl)-1-(oxane-2-carbonyl)piperidine
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-(3-chlorobenzoyl)-1-[(4-methoxyphenyl)methyl]piperidine
5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(1-methylcyclohexanecarbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
1-(1-benzylpiperidin-4-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
2,5-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
2-cyclopropyl-N-methyl-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,6-dihydropyrimidine-5-carboxamide
1-(furan-2-ylmethyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]piperidine-4-carboxamide
2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
{5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]furan-2-yl}methanol
2-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-benzyl-N3-[1-(6-methoxynaphthalen-2-yl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-chloro-2-{[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}phenoxy)acetic acid
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-{4-[(3,4-difluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-methyl-1,4-diazepane
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(quinolin-6-ylmethyl)propanamide
1-(3-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
1-cyclopentanecarbonyl-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
N,N-diethyl-1-[(1s,4s)-4-(2,3-dihydro-1-benzofuran-2-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidine-3-carboxamide
2-cyclopropyl-5-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-4-methylpyrimidine
1-(3-chlorobenzenesulfonyl)-N-(3,4-difluorophenyl)piperidin-3-amine
2-(3-chlorophenoxy)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}propanamide
5-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-4-amino-1-[2-(2-oxoazepan-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 2-[8-(2-methylpropyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-(2-{2-azaspiro[4.4]nonan-2-ylmethyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]quinoline