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N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)acetamide
N-benzyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-fluoro-2-methoxy-N-methylbenzamide
(3S,4R)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(benzyloxy)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
N-[(1-methylpyrrolidin-3-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-(2-methyl-6-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-yl}pyrimidin-4-yl)morpholine
1-cyclopentyl-N-[2-(N-methylmethanesulfonamido)ethyl]-5-oxopyrrolidine-3-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
{2-[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}urea
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
2-{4-[6-(dimethylamino)pyrimidin-4-yl]phenyl}-2-methylpropanenitrile
1-(3-chlorophenyl)-4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}piperazin-2-one
5-(methoxymethyl)-N-({7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
(2E)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-4-yl)prop-2-enamide
2-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N-ethyl-N-methylpyrimidin-4-amine
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(2-methoxyphenyl)methyl]piperidine
(3aS,6aS)-2-[(3-chloro-5-fluorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-methoxyethyl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)propanoic acid
N-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-[1-(cyclohexylmethyl)-1H-1,2,3-triazol-4-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
1-(3-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-5-oxopyrrolidine-3-carboxylic acid
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
4-methyl-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pentanamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-2-yl)propan-1-one
4-chloro-N-(3-hydroxypropyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl]methanol
2-(dimethylamino)-N-{3-[({1-oxaspiro[4.5]decan-3-yl}carbamoyl)amino]phenyl}acetamide
5-(2,5-dimethylfuran-3-yl)-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-1,2,4-triazine
N-[(2R,3R)-2-methoxy-1'-[3-(2-oxopiperidin-1-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1,2,5-tetramethyl-1H-pyrrole-3-carboxamide
4-(9H-fluoren-9-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-2-methyl-1,4-diazepan-5-one
2-[(3,5-difluorophenyl)methyl]-8-(3-methoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
4-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]pyridine
5-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)furan-2-carboxamide
N-cycloheptyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 1-benzyl-5-(2,6-dimethylpyrimidine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
8-[2-(ethylsulfanyl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-methoxyquinolin-3-yl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
ethyl({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylate
1-[3-(4-chlorobenzoyl)piperidin-1-yl]-4-phenylbutane-1,4-dione