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N-cyclopropyl-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazine-2-carboxamide
N-(2-acetylphenyl)-3-(thiomorpholin-4-yl)propanamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-[(4-methoxyphenyl)methyl]-1H-1,3-benzodiazole
[4-fluoro-7-(1,3-thiazol-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
(3R,4R)-4-amino-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidin-3-ol
1-methyl-2-(morpholin-4-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-chlorophenyl)methyl]-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(6-methylquinoline-4-carbonyl)piperidin-4-yl]propanamide
4-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)piperidin-2-one
[(4-cyclopropyl-5-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
6-{[4-(diethylamino)phenyl]methyl}-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-(propan-2-yloxy)ethan-1-one
4-{5-[(2,4-dimethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine
N-(1-{7-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
methyl 3-{[5-(3-chlorothiophene-2-carbonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-[3-(4-{[2-(2,3-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-(pyridin-3-yl)propanamide
1-methyl-9-(prop-2-en-1-yl)-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
7-[(4-fluorophenyl)methyl]-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-cyclopropyl-6-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
5-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(3S,4S)-1-(2-methylpyridine-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(3R)-4-[(2-methoxy-3,5-dimethylphenyl)methyl]morpholine-3-carboxylic acid
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
4-(4-fluorophenyl)-N-methyl-4-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
2-[4-(1-benzothiophen-3-yl)-2-(pyrrolidin-1-ylmethyl)phenoxy]-N-[(3,4,5-trimethoxyphenyl)methyl]acetamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
3-acetamido-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(2-methoxyphenoxy)piperidine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2,4-dimethyl-1,3-oxazole-5-carboxamide
N-{[7-(dimethyl-1,3-thiazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amine
4-methoxy-6-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidin-2-amine
2-cyclobutyl-5-fluoro-1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
3-{5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
[1-(2-chlorobenzoyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-[1-(methoxymethyl)cyclopropyl]-3-methylurea
2-{5-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(1S,5R)-6-[(2-methoxy-3,5-dimethylphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5,6-dimethylthieno[2,3-d]pyrimidine
2-(1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}pyrrolidin-3-yl)benzoic acid
5-{4-hydroxy-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N4-cyclopropyl-6-(4-{[2-(methylamino)pyridin-3-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine