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2-{4-[(2,6-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
N-(furan-2-ylmethyl)-1,4,6-trimethyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-acetyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)thiophene-2-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
9-(5-chloropyridin-2-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-hexyl-8-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{2-methoxy-4-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamido]phenyl}-3-methylbutanamide
N-({8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
(1R,5R)-6-propyl-3-(pyridazine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-[(4-fluorophenyl)methyl]-2-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,7-diazaspiro[4.5]decane
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]acetamide
methyl 3-{2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetamido}azepane-1-carboxylate
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methoxyphenyl)propanamide
3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
N-benzyl-3-propoxypiperidine-1-sulfonamide
3-(2-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
[4-(2-phenylethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl]methanol
N-methyl-3-(piperidine-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]pyrazine-2-carboxamide
5-ethoxy-N-[(1-ethylpiperidin-3-yl)methyl]furan-2-carboxamide
1-(4-chlorobenzoyl)-3-(2-methoxybenzoyl)piperidine
5-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
2-benzyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1,3-thiazole-4-carboxamide
2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
3-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamido]propanoic acid
methyl(naphthalen-1-ylmethyl)[(4-{[1-(pyridine-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
2-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)benzoic acid
3-(but-2-yn-1-yl)-5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-(3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
(3R,9aR)-3-benzyl-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{1-[2-(4-chloro-2-methylphenoxy)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]ethan-1-one
4-[7-(oxane-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
(2S)-2-({[3-(pyridin-2-ylmethoxy)phenyl]methyl}amino)propanamide
3-(dimethyl-1,3-thiazol-5-yl)benzoic acid
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepane
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
3-[(4-fluorophenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(cyclopropylmethyl)-3-hydroxy-3-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}piperidin-2-one
1-(propan-2-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]piperidine-4-carboxamide
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-4-(piperidin-3-yl)benzamide
1-(cyclopropylmethyl)-4-(2-methylpyrimidine-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-fluoroethyl)benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
3-{2-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
ethyl 3-[(2-fluorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate