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2-fluoro-N-{[8-(1-phenylcyclopropanecarbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
7-chloro-3,5-dimethyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-benzofuran-2-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)but-2-ynamide
3-[(cyclopentylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
1-(2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
2-(2-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
methyl (2S,4S)-1-[(2,5-dimethylphenyl)methyl]-4-(2-methoxybenzamido)pyrrolidine-2-carboxylate
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
1-cyclopropanecarbonyl-N-[2-(pyrazin-2-yl)ethyl]piperidine-4-carboxamide
5-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
methyl 3-(2-cyclopentylacetyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl (2S,4S)-4-(3-chlorobenzamido)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1-benzofuran-2-carboxamide
1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(furan-3-carbonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N4-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine
2-(4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
1-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-{2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1,3-benzothiazole-5-carboxamide
3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-methylbenzoic acid
N-(2-{7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
6-(2-methylbutyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[5-(5-ethylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-(1-benzothiophen-2-ylmethyl)-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}quinoline-3-carboxamide
5-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-2-(propan-2-yl)pyrimidine
3-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
(3S,4R)-3-benzyl-1-(5-chloropyridin-2-yl)-4-methylpiperidin-4-ol
4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]pyrrolidin-3-ol
2-(2-chloro-4-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
4-[7-(pyridine-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyridin-1-ium-1-olate
N-[(3,5-dimethoxyphenyl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
1-cyclopropyl-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
(2R)-2-amino-3-(4-chlorophenyl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
2-ethyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide
4-hydroxy-1-(3-methyl-1-benzothiophene-2-carbonyl)piperidine-4-carboxylic acid
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-methylpentanamide
4-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
3-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-methyl-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(pyridin-2-yl)piperidin-4-ol