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(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
5-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methylpyridine
1-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cyclopropane-1-carboxamide
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-({[4-(propan-2-yloxy)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-4-(1-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1,3-thiazole
7-[(4-chlorophenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-(3-chlorophenyl)-3-(1-ethoxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
ethyl 4-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1H-pyrazole-3-carboxylate
1-(carbamoylmethyl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)piperidine-3-carboxamide
N,N-dimethyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)azepan-4-amine
ethyl 4-(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazole-7-carbonyl)piperazine-1-carboxylate
1-[4-(3-chlorophenoxy)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
8-(5-fluoropentyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(5-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
3-{benzyl[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}-2-methylpropan-1-ol
1-(oxane-2-carbonyl)-4-(2-phenylethyl)piperazine
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-acetyl-6-methyl-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl)(quinolin-8-ylmethyl)amine
N-[3-(1H-imidazol-1-yl)propyl]-6-oxo-N-(pyridin-4-ylmethyl)-1,6-dihydropyridine-2-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(oxan-4-yl)-1,3-oxazole-4-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidine-4-carboxylic acid
N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
(4aS,8aR)-6-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-1-(2-aminoethyl)-decahydro-1,6-naphthyridin-2-one
N-{[3-(3-methyl-1H-pyrazol-4-yl)phenyl]methyl}acetamide
(2E)-N-({7-[3-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
(4-{[1-(3-methylphenyl)-1H-pyrrol-2-yl]methyl}morpholin-2-yl)methanamine
1-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-3-phenylpropan-1-one
2-(3-methoxypropyl)-4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N,N-dimethyl-4-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}-4-oxobutanamide
3-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]phenol
ethyl 4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxylate
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
3-{[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl](propan-2-yl)amino}propanamide
5-(4-methylpiperidine-1-carbonyl)-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
3-methoxy-1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
4-chloro-5-{[4-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
1-methyl-5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
6-chloro-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
1-cyclopentyl-4-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperazin-2-one
methyl({[5-(pyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(methylamino)propan-1-one
3-phenyl-5-(thiomorpholine-4-sulfonyl)-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]benzamide