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N-[(2S)-1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-methyl-1-oxopentan-2-yl]acetamide
2,4-dibenzyl-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 3-[2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamido]propanoate
1-(2-chlorophenyl)-4-[2-(pyridin-2-yl)acetyl]piperazin-2-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)acetamide
3-{1-[2-(4-ethoxyphenyl)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-ethylphenyl)-1H-pyrazole-5-carboxamide
2-[2-(2,5-dimethylphenyl)phenoxy]propanamide
2-[({4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)methyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-[(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
ethyl 2-{4-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]morpholin-3-yl}acetate
5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
6-(2-ethoxypyridin-3-yl)-1,3-benzothiazole
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-fluoro-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 3-{9-methoxy-7-oxo-10-[(thiophen-2-ylmethyl)carbamoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-3-carbonyl}benzoate
N-[(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-3-phenylpropanamide
N2,N2,5,6-tetramethyl-N4-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-2-carbonitrile
5-{2-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
2-{[4-(3-acetylphenyl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carboxamide
N-benzyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1R,3S,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]acetamide
1-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(pyridin-2-yl)propan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
1-cyclopropyl-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
7-chloro-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-9-oxo-9H-fluorene-1-carboxamide
N-(4-fluorophenyl)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-amine
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
3-(2-methylpropyl)-1-[(3-methylpyridin-2-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-phenyl-1H-pyrazole-4-carboxamide
1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylpiperidin-4-yl)piperidine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(morpholin-4-yl)pyridine-3-carboxamide
5,5-dimethyl-1-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
[(3S,5R)-1-benzoyl-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]propan-1-one
1-(2-methoxyethyl)-N-methyl-N-[3-(phenylsulfanyl)propyl]pyrrolidine-3-carboxamide
(1S,5S)-3-[(3-methyl-1-benzofuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
8-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
3-(1H-1,3-benzodiazol-1-yl)-N-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
5-(2-methoxy-4-methylphenoxymethyl)-N-[2-(methylamino)ethyl]-1,2-oxazole-3-carboxamide