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5-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,2-oxazinane
1-(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)piperidine
(2S,4R)-N-ethyl-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazol-1-yl}acetamide
(3R,7S,8aS)-7-{[(5-chlorothiophen-2-yl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2,3-dimethyl-N-[1-(thiophen-3-yl)propan-2-yl]quinoxaline-6-carboxamide
1-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
2-methoxy-6-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
N-cyclopropyl-4-(2-ethoxyphenyl)benzamide
3-({[(1-ethylcyclopropyl)methyl]amino}methyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
7-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2,3-dimethyl-1H-indole
2-[5-(methanesulfonylmethyl)pyridin-2-yl]benzonitrile
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)-N-methylacetamide
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[2-(4-chlorophenyl)ethyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
8-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(4S)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-{[3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-phenoxyacetamide
4-(2-butyl-1,3-benzoxazole-5-carbonyl)piperazin-2-one
N,1-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]azepane-2-carboxamide
4-(3-chlorothiophene-2-carbonyl)-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-(1-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
methyl 4-[({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)methyl]benzoate
2-({2-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(1-hydroxybutan-2-yl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
2-methyl-4-phenyl-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecane
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
2-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrazine
7-[ethoxy(phenyl)methyl]-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-amino-4-{4-[(dimethylamino)methyl]thiophen-2-yl}-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
[(2-chlorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-[1-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1H-1,2,3-triazol-4-yl]piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-ethyl-3-(piperidin-3-yl)-1-(pyrimidin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-N-({7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)butanamide
N-{[1-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-3-yl]methyl}acetamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(thiophene-2-carbonyl)piperidine
2-{5-[(2S)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-ethyl-8-[(2E)-3-phenylprop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methoxy-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidin-1-yl)pyridazine
N-[(3,4-dimethoxyphenyl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methylpropanamide
N6-methyl-N6-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-9H-purine-2,6-diamine
8-methoxy-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(3-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}phenyl)-2-methylbut-3-yn-2-ol