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1-(2,3-dihydro-1H-inden-2-yl)-4-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-1,4-diazepane
dimethyl[(3-methylphenyl)({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl})methyl]amine
{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-sulfonamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[1-(4-fluorophenyl)ethyl]amine
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-(3-methylphenoxymethyl)piperidine
N2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methylpyrimidine-2,4-diamine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
[(3S,5R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
4-hydroxy-1-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)piperidine-4-carboxamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
5-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R,3R)-1'-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}-2-(methylsulfanyl)pyrimidine
N-(2-methoxy-2-methylpropyl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-4-hydroxypiperidine-4-carboxylic acid
2-(3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidin-1-yl)pyridine
{4-[1-(2-methylbenzoyl)piperidine-4-carbonyl]-1,4-oxazepan-6-yl}methanol
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{1-[(1,3-dimethylpyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
5-(1-carbamoylcyclopropanecarbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(4aR,8aR)-2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-acetamido-3-methylbutanamide
methyl 5-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-methoxypiperidine
methyl 1-{2-hydroxy-3-[4-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
5-(4-chlorophenyl)-N-(pyridin-4-ylmethyl)-1,2,4-triazin-3-amine
N-(1-{1-[(dimethylcarbamoyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}propan-2-yl)furan-2-carboxamide
5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyrazin-2-ol
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
N-[3-(2-phenylacetamido)phenyl]oxolane-3-carboxamide
N-(1H-indol-2-ylmethyl)-3-(4-methylpiperazin-1-yl)propanamide
(4aS,8aR)-1-(3-aminopropyl)-2-oxo-N-(2-phenylethyl)-decahydro-1,6-naphthyridine-6-carboxamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(2-oxoazepan-1-yl)acetamide
6-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile
N-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]cyclobutanecarboxamide
2-{[(4-cyanooxan-4-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[2-(4-chlorophenyl)ethyl]-N-(oxan-4-yl)-6-oxopiperidine-3-carboxamide
5-(1-benzofuran-2-yl)-3-[4-(pyridin-4-yl)piperidin-1-yl]-1,2,4-triazine
(5S,9aS,9bS)-5-(4-fluorophenyl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one