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2-ethyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
5-(2,6-difluorophenoxymethyl)-N-[1-(4-fluorophenyl)propyl]-1,2-oxazole-3-carboxamide
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-(5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-[(3-fluorophenyl)methyl]-4-[(6-phenylpyridin-3-yl)methyl]piperazine
N-ethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
1-(3,4,5-trimethoxyphenyl)-1H-pyrazolo[3,4-b]pyridine
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]benzonitrile
4-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridine
1-(cyclohexylmethyl)-N-methyl-5-[4-(thiophene-2-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-hydroxy-3-methylphenyl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(3-phenylpropyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2R)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}oxolane-2-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-methyl-4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
7-(propan-2-yl)-2-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2,5,6-trimethyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
N-(furan-2-ylmethyl)-2-propyl-N-(thiophen-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-[4-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)piperazin-1-yl]ethan-1-ol
N-(1-{7-[2-(2,5-difluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
2-methyl-1-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}-4-phenylpiperazine
3-(4-ethyl-1H-pyrazol-5-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(1-phenylcyclohexyl)methyl]amine
N-methyl-N-[(1-phenyl-1H-1,2,4-triazol-5-yl)methyl]cyclopentanamine
N-[3-(4-{[3-(furan-2-yl)-3-phenylpropyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
1-[2-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-ol
(2S,4S)-4-amino-1-(isoquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-(4-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
methyl (2S)-1-{9-methoxy-3-[(2-methyl-1H-indol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}benzamide
N-[4-({[(1-methyl-1H-imidazol-2-yl)methyl](propyl)carbamoyl}methoxy)phenyl]propanamide
3-[2-(2-cyclopropyl-1H-imidazol-1-yl)ethyl]-1,3-oxazolidin-2-one
2-[3-(2-methoxyphenoxy)azetidin-1-yl]quinoline-4-carboxylic acid
1-(4-methoxyphenyl)-6,6-dimethyl-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
(2S)-2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)-3-phenylpropanamide
4-ethyl-3-{1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
ethyl 1-benzyl-5-(1-methoxypropan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(dimethylamino)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[4-(morpholine-4-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-[(dimethylamino)methyl]-1-[(5-methoxy-1H-indazol-3-yl)methyl]pyrrolidin-3-ol
methyl 4-({[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}methyl)benzoate
2-chloro-N-(1-cycloheptylpiperidin-3-yl)-4-fluorobenzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione