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(2S)-2-amino-1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-cyclohexylethan-1-one
4-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1λ6-thiomorpholine-1,1-dione
{2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}urea
8-methoxy-N-[2-(3-methoxyphenoxy)ethyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl N-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}carbamate
N-cyclohexyl-1,5-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
4-(3,4-difluorobenzoyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
3-({1-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
5-methyl-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}pyrazine-2-carboxamide
4-(1H-imidazol-2-yl)-1-[(2S)-1-methanesulfonylpyrrolidine-2-carbonyl]piperidine
N,N-diethyl-1-{5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-amine
methyl 3-[5-(methoxymethyl)furan-2-carbonyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
1-(piperidin-1-yl)-3-[4-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-(cyclopropylmethyl)-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl 3-[3-(4-methoxyphenyl)propanoyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclooctyl-2-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}acetamide
2-methyl-8-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
4-(4-methylphenoxy)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
3-(2-amino-1,3-thiazol-4-yl)-N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]propanamide
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[(4-chlorophenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3-(trimethyl-1H-pyrazol-1-yl)propanamide
4,6-dimethyl-3-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N4-[3-(2-fluorophenyl)propyl]-2-methylpyrimidine-4,6-diamine
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
N-tert-butyl-2-(4-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}phenoxy)acetamide
4-(1-ethyl-1H-imidazol-5-yl)-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(1H-1,3-benzodiazol-1-yl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-4-carboxylic acid
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(methylsulfanyl)propanamide
(3E)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pent-3-enamide
2-(6-methoxy-1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-2,5-dihydro-1H-pyrrole-2-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-ethyl-3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
N-{[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenoxyacetamide
methyl 7-oxo-3-(4-oxopentanoyl)-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]pyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-3-methoxy-N-[(2-methylphenyl)methyl]propanamide
1-{2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}piperidin-2-one
4-chloro-1-methyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(furan-2-yl)-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
7-(5-chloropyridin-2-yl)-4-[(2-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3-oxa-9-azaspiro[5.5]undecane