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N-[(2S,4R,6R)-2-(3-methyl-1-benzothiophen-2-yl)-6-(propan-2-yl)oxan-4-yl]acetamide
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(oxane-4-carbonyl)piperidine
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
N-({1-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]piperidin-3-yl}methyl)-4-fluorobenzamide
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-ethyl-2,6-dimethylpyrimidine
2-(3-fluorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-[2-(3,4-difluorophenyl)ethyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
N-cyclopentyl-4-(4-{[2-(1H-indol-3-yl)ethyl]amino}piperidin-1-yl)benzamide
3-[1-(pyridine-3-sulfonyl)piperidin-3-yl]benzoic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-7-fluoro-1,2,3,4-tetrahydroisoquinoline
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
(3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-oxopropyl)urea
1-(1,3-oxazole-5-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
ethyl 1-(3-methylbenzoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,3-thiazole-5-carboxamide
3-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1,4-dithiepan-6-amine
(3aR,6aR)-2-cyclopentanecarbonyl-5-(5-ethyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3S,5R)-5-[(dimethylamino)methyl]-1-(2,6-dimethylpyridine-4-carbonyl)piperidin-3-yl]methanol
3-(2-ethoxypyridine-3-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
N-[4-(propan-2-yl)phenyl]-1-(quinoxaline-6-carbonyl)piperidin-3-amine
(2S)-1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-2-phenylethan-1-one
4-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N4-methyl-6-(morpholin-4-yl)-N4-(thiophen-3-ylmethyl)pyrimidine-2,4-diamine
ethyl 5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3aR,6aR)-2-(3,5-dimethylbenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-4-yl)-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
3-(methylsulfanyl)-1-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
1-(4-ethoxyphenyl)-2-(3-methylfuran-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
3-[2-(2-methylpropanesulfonyl)ethyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(4-methylphenoxymethyl)piperidine
1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidine
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
1-methyl-2-oxo-8-(5-phenylpentanoyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-ethyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidin-4-amine
7-fluoro-2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-4-carboxamide
1-[(2S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane