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1-(2-methyl-5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
(1r,4r)-4-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexane-1-carboxamide
3-{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-(1-ethyl-1H-pyrazol-4-yl)-2-(furan-2-yl)pyrrolidine-1-carboxamide
N-benzyl-N-(cyclopropylmethyl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
5-[3-(1H-pyrazol-5-yl)phenyl]furan-2-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-(2-fluoroethyl)-3-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]sulfonyl}benzamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{3-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]phenyl}ethan-1-one
4-(6-methoxypyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[(4-fluorophenyl)methyl]-3-methyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
3-[3-cyclopropyl-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
N-propyl-N-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-propyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[2-(2-oxopiperidin-1-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-{1-[(4-methoxynaphthalen-1-yl)methyl]azetidin-3-yl}pyridine
ethyl 3,5-dimethyl-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-pyrrole-2-carboxylate
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-tert-butyl-3-[(cyclohex-3-en-1-ylmethyl)amino]-5-(4-methyl-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methyl-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-(pyridin-2-ylmethyl)piperidin-3-amine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carbonyl}azepane
8-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
(1S,5R)-3-(1-tert-butyl-1H-pyrrole-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(1,3-benzothiazol-2-yl)-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
9-methoxy-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4S)-3-hydroxy-4-(4H-1,2,4-triazol-4-yl)-1λ6-thiolane-1,1-dione
4-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H-chromene-2-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-1,2-dihydroisoquinolin-1-one
1-(3-butoxyphenyl)-3-[2-(1H-pyrazol-4-yl)ethyl]urea
methyl 5-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}furan-2-carboxylate
(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-7-[(thiophen-2-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-{1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
N-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-1-(4-chlorophenyl)cyclopropane-1-carboxamide
N-[3-(pyridin-2-yl)propyl]-6-[2-(pyridin-2-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
6-fluoro-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
3-{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
methyl (2S,4S)-4-acetamido-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxylate
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-ethenylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-3-ethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
3-{1-[(3-chlorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
7-[(2-phenylphenyl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one