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1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
N-[(2R,3R)-1'-[(2,5-dimethylphenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-(dimethylamino)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
4-(dimethylamino)-N-[4-(2-fluorophenoxy)phenyl]azepane-1-carboxamide
9-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]acetamide
2-{[4-(2-methoxyquinolin-3-yl)phenyl]sulfanyl}acetamide
N-ethyl-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}acetamide
(1S,6R)-9-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N5-(1-ethylpiperidin-4-yl)-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
2-(2,4-dichlorophenoxy)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
2-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
(4aS,8aR)-6-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methylbenzamide
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2,2-bis(prop-2-en-1-yl)piperidine
1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
2-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2-ethyl-4-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
N-(2-methoxyethyl)-N-methyl-5-phenyl-1,2,4-triazin-3-amine
N-ethyl-5-[3-(phenoxymethyl)piperidine-1-carbonyl]pyrimidin-2-amine
(2R,3R,6R)-5-(furan-2-ylmethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(4-fluorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-{[methyl({[1-(2-methylpropyl)piperidin-4-yl]methyl})amino]methyl}benzene-1,2-diol
2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1,2-benzothiazol-3-one
2-(3-methoxypropyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
8-fluoro-2-({[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)quinolin-4-ol
(3R,4S)-1-cyclohexyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N,N-dipropyl-1,3-oxazole-4-carboxamide
2-{5-[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol
(4aR,7aS)-1-benzyl-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-chloro-4-fluoro-5-methylphenyl)-1-[(1-hydroxycyclohexyl)methyl]urea
2-({5-[2-amino-3-cyano-6-(trimethyl-1H-pyrazol-4-yl)pyridin-4-yl]pyrimidin-2-yl}amino)acetic acid
N-{[3-methyl-7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-2-yl)acetamide
N-methyl-1-[(2-methylphenyl)methyl]-N-[(4-phenoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(ethylamino)-N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
3-({1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-5,5-dimethylimidazolidine-2,4-dione
2-(2-butyl-1H-imidazol-4-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
3-(3-hydroxyquinoxalin-2-yl)-1-[(2S)-4-methyl-2-phenylpiperazin-1-yl]propan-1-one
4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methoxypyrimidine
3-hydroxy-3-({[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
2-{2-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazine
2,2-dimethylpropyl 2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-[(4-fluorophenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)thiophene-2-carboxamide
5-(2-methoxyacetamido)-1-methyl-N-(3-phenylpropyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide