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N,1,3-trimethyl-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
N-[(5-methylfuran-2-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
(3S)-1-ethyl-4-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-methylpiperazin-2-one
(1S,5R)-6-[(5-methylthiophen-2-yl)sulfonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
6-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1,3-benzothiazole
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
5-chloro-N,4,6-trimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
9-methoxy-4-(4-methoxybenzenesulfonyl)-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
methyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-[(4-butoxyphenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-(3-methoxyphenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
3-(1-{[1-(2-amino-5-chloro-6-methylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N'-{1-azabicyclo[2.2.2]octan-3-yl}-N-cyclopentylbutanediamide
2-{5-[1-(4-methoxyphenyl)cyclopentyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-(2-chlorophenyl)-N-[2-(dimethylsulfamoyl)ethyl]furan-2-carboxamide
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(3-phenylprop-2-ynoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(2-ethoxyethoxy)-4-[(E)-2-(furan-2-yl)ethenyl]-1,2,3,4-tetrahydroquinolin-2-one
(2S,4R)-4-{[(2,5-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-(adamantan-1-yl)-N-(3-ethoxy-2-hydroxypropyl)-4-hydroxypyrimidine-5-carboxamide
(2S)-2-amino-N-benzyl-N-(1,3-thiazol-2-ylmethyl)-3-(1,3-thiazol-4-yl)propanamide
(5S)-5-({[(1-methyl-1H-imidazol-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)but-3-enamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(pyrrolidin-1-yl)benzamide
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
14-(1-ethyl-1H-1,2,4-triazol-5-yl)-2,17-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3,5,7,11,13(18)-hexaen-16-one
6-propyl-2-[2-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(1,4-oxazepane-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
2-amino-4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)quinazoline-6-carboxylic acid
N,N-dimethyl-2-{3-[3-(quinolin-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1,2-oxazole
{3-[(2,4-difluorophenyl)methyl]-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl}methanol
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-6-(2-methoxyethyl)-3-[4-(piperidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
ethyl 4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazine-1-carboxylate
2-amino-N-benzyl-N-methyl-1,3-benzothiazole-5-carboxamide
1-(2-chlorophenyl)-4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
N-methyl-N-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl)methanesulfonamide
4-{pyrazolo[1,5-a]pyridin-7-yl}pyrimidin-2-amine
6-methyl-4-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-cyclopropyl-3-[1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-4-yl]propanamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrazine-2-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
1-methyl-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-imidazole-5-carboxamide
(3S,4R)-N-[(4-chlorophenyl)methyl]-3-[(dimethylcarbamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carboxamide