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1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-(2-chloro-4,5-difluorophenyl)ethan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,3-benzothiazole-6-carboxamide
3-{4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl}propanamide
N-cyclopropyl-N-(2-phenyl-1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}ethyl)furan-2-carboxamide
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)pyrazine-2-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
[(2,3-dimethoxyphenyl)methyl][(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
3-ethoxy-1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
2-[(4-chlorophenyl)methyl]-8-(morpholine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-{2-[3-(hydroxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
7-{[2-methyl-5-(1,2-oxazol-5-yl)furan-3-yl]sulfonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
4-[2-(morpholin-4-yl)butanoyl]-1-phenylpiperazin-2-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
5-methoxy-3-methyl-2-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}-1H-indole
1-{5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
7,7-dimethyl-2-[2-(oxolan-3-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-1-cyclohexyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
1-[(2S)-2-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}pyrrolidin-1-yl]ethan-1-one
{1-benzyl-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
1-[(2-chlorophenyl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
3-cyclopentyl-1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}propan-1-one
(2E)-N-{[7-(5-acetylthiophene-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(1-phenylpiperidin-4-yl)acetamide
ethyl 5-benzoyl-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
7-(1,3-benzothiazol-2-yl)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[phenyl(pyridin-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(dimethylamino)butyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
2-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)amino)-N-methylpropanamide
2-{[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
5-{1-[(6-phenoxypyridin-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methylthiophen-2-yl)methyl]benzamide
N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(thiophen-3-ylmethyl)acetamide
7-[(3-methylphenyl)methyl]-2-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
(1R,7S)-3-cycloheptyl-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2-phenylpyrimidine
2-(3-{1-[(2R)-2-hydroxy-2-phenylethyl]-1H-pyrazol-3-yl}phenyl)pyridine-4-carbonitrile
7-(cyclobutylmethyl)-2-(1,3-thiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-methoxy-5-{2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}pyridine