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3-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
6-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(1S,5R)-3-methyl-6-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-1-(azepane-1-sulfonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(1S,6R)-3-methyl-9-(1,8-naphthyridine-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[2-(furan-2-yl)ethyl]-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-4-carbonitrile
5-oxo-1-[4-(propan-2-yl)phenyl]-N-(pyrimidin-4-ylmethyl)pyrrolidine-3-carboxamide
2,6-dimethoxy-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
1-methyl-N-[(8-{[4-(2-methylpropyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N'-cyclopentyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanediamide
3-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]propanamide
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(thiophen-3-yl)pyridine-3-carboxamide
N-[3-(3-methoxypyridin-2-yl)phenyl]acetamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(3-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
4-(5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-yl)morpholine
N-(furan-2-ylmethyl)-3-(1H-indole-6-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(furan-2-yl)ethyl]-7-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
methyl 3-{[(4-methyl-1,3-oxazol-5-yl)formamido]methyl}-5-(2-phenylacetamido)benzoate
N-ethyl-6-methoxy-N-(oxan-4-ylmethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
1-cyclopentyl-3-methyl-5-(5-methylfuran-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(thiophene-2-sulfonyl)-decahydro-1,6-naphthyridin-2-one
7-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
6-(4-chlorophenyl)-N-(2,5-dihydroxy-2-methylpentyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(2-methylpropyl)piperidin-3-yl)methanol
(4aS,8aS)-2-(3-chloro-4-fluorobenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
(3R,9aR)-8-[(2-chlorophenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-cycloheptylpiperidin-3-yl)-2-(morpholin-4-yl)benzamide
4-[1-(2,5-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]piperidine
2-butyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
1-methyl-1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2,6-difluorophenyl)methyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(1-benzofuran-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-[benzyl(methyl)amino]-3-[5-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
3-cyclopropyl-5-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
5,7-dimethyl-2-(pyrimidin-5-yl)quinolin-8-ol
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
3-chloro-4-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyridine
(3aS,6aS)-2-[(2-methylpyridin-3-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-[4-({[1-(2-fluorophenyl)piperidin-4-yl]carbamoyl}amino)phenyl]-N-methylacetamide
4-[1-benzyl-5-(2-chloropyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-methyl-8-{thieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide