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3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[4-(pyridin-2-ylmethoxy)phenyl]urea
5-(2H-1,3-benzodioxol-5-yl)-3-(ethoxymethyl)-1-[2-(1H-imidazol-5-yl)ethyl]-1H-1,2,4-triazole
2-(4-{[4-(methylamino)piperidin-1-yl]methyl}phenyl)-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
4-(2-methoxyphenyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2,6-dihydroxybenzamide
N-[2-(4-methoxyphenyl)ethyl]-4-methyl-N-[(1-methylpiperidin-4-yl)methyl]pyrimidine-5-carboxamide
3-[1-methyl-2-(methylcarbamoyl)-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-6-carbonyl]piperidine-1-carboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-(1-propylpiperidin-4-yl)imidazolidine-2,4-dione
1,6-dimethyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-2-[1-(thiophene-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
5-(1H-pyrazol-3-ylmethyl)-2-[2-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-(azocan-1-yl)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-ol
4-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-imidazole-5-carboxamide
5-methanesulfonamido-N-[2-(2-methoxyphenyl)ethyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-(4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-ethyl-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-propanoylphenoxy)acetamide
N-methyl-3-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}benzamide
2-cyclohexyl-5-{1-[2-(propan-2-yloxy)ethyl]-1H-imidazol-2-yl}pyrimidine
6-(dimethylamino)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
2-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-N-methylacetamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
2-(2-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
4-(1H-imidazol-1-yl)-1-(1-methyl-1H-indole-3-carbonyl)piperidine-4-carboxylic acid
2-(4-methylphenoxymethyl)-N-(4H-1,2,4-triazol-4-yl)furan-3-carboxamide
5-methyl-5-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
3-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
(9aS)-2-[2-(benzyloxy)ethyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
1-(2-benzylmorpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
2-({1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
1-methanesulfonyl-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
4-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-(cyclopropylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
6-cyclopentyl-N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenyl]ethan-1-one
2-(dimethylamino)-1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(3-methylphenyl)ethan-1-one
N-(2-methoxyethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1H-1,2,4-triazole-5-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentylquinoline-2-carboxamide
3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
8-fluoro-2-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)quinolin-4-ol