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N-(2,2-dimethyloxan-4-yl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-N-methylthiophene-2-carboxamide
1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
6-[2-(4-fluorophenyl)morpholine-4-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
methyl 4-{[3-(morpholin-4-yl)piperidine-1-carbonyl]amino}benzoate
1-ethenyl-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2,4-difluorophenoxy)-1-(2,3-dihydro-1H-isoindol-2-yl)ethan-1-one
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2-(1-methylpiperidin-2-yl)acetamide
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}sulfonyl)morpholine
1-(azocan-1-yl)-3-(4-{[(3-ethoxypropyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
(3S,9aR)-3-[(benzyloxy)methyl]-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3,5-dimethyl-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-1,2-oxazole-4-sulfonamide
2-methyl-6-[1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]pyrimidin-4-ol
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
1-(4-{4-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]piperazin-1-yl}phenyl)ethan-1-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{[2-(2-carboxyethyl)piperidin-1-yl]methyl}benzoic acid
2-fluoro-N-{3-[(3R)-3-hydroxypyrrolidin-1-yl]-3-oxopropyl}benzamide
3-{2-[(3R)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
3-methyl-N-{3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]phenyl}benzamide
ethyl 2-[1-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)cyclohexyl]acetate
5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
4-[2-(pyrrolidin-1-yl)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]propanamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-methyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-2-phenylpiperazine
1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline
N-[1-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(pyridin-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3S)-3-ethylmorpholin-4-yl]propan-1-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-3,4-dimethoxybenzamide
1-[(1s,4s)-4-aminocyclohexyl]-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[2-(4-ethylpiperazin-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-[(3R,4S)-1-[(5-chlorothiophen-2-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-2-methoxyacetamide
2-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
1,5-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
N-(4-chloro-3-methoxyphenyl)-2-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-methylphenol
3-(oxolan-3-yl)-5-[3-(1H-1,2,4-triazol-3-yl)phenyl]-1H-1,2,4-triazole
methyl(1,2-oxazol-3-ylmethyl)[(4-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-fluorophenyl)benzamide
methyl 4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)thiophene-2-carboxylate
2-(4-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one