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2-(3-hydroxyphenyl)-N,N-dimethylbenzamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-propylpiperidine-3-carboxamide
2-cyclopentyl-1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
dimethyl({[(1R,5S,6S)-3-(3-phenyl-1,2-oxazole-5-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
(2S)-N-[3-(1H-pyrazol-1-yl)phenyl]-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidine-2-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(1H-imidazol-1-ylmethyl)piperidine
5-({2-cyclopropyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(2-methylphenyl)-4-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]piperazine
methyl 3-{[1-(4-methylquinazolin-2-yl)piperidin-4-yl]formamido}propanoate
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-hydroxy-N-methylpyrazine-2-carboxamide
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(oxan-4-yl)sulfamoyl]-N-(pyridin-3-yl)benzamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-{[7-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
propyl 7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,7-diazaspiro[4.5]decane-2-carboxylate
N,N-diethyl-2-[4-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1H-1,2,3-triazol-1-yl]acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-7-methoxyquinolin-2-yl]-4-[2-(dimethylamino)ethyl]-1,4-diazepan-5-one
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
N-(2-fluorophenyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
2-methyl-4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]phenol
1-[(4-chlorophenyl)methyl]-4-(1-methylpiperidine-2-carbonyl)piperazine
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(1H-indol-1-yl)propan-2-yl]propanamide
1-methyl-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}urea
4-ethyl-3-(1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,3R,6R)-5-cyclopentanecarbonyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1-benzofuran-2-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(1-benzofuran-2-ylmethyl)[(1-ethylpyrrolidin-3-yl)methyl]methylamine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
4-({1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(1-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
7-(5-chloropyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(dimethylamino)-2-(3-fluorophenyl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propyl-5-[1-(2,4,5-trifluorobenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
1-[(benzylcarbamoyl)methyl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(4-methoxyphenyl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[(1-phenylcyclohexyl)methyl]piperidin-4-amine
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrrol-2-yl)pyridine
2-(2H-1,3-benzodioxol-5-yl)-1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-(3-phenylpropyl)-3-(pyrrolidin-1-ylmethyl)piperidine
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
N4-(1-cyclopentanecarbonylpiperidin-4-yl)-6-(propan-2-yl)pyrimidine-2,4-diamine
N-[2-(1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(4-{[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl}piperazin-1-yl)ethan-1-ol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
propyl 4-{[3-(3-fluorophenyl)phenyl]carbamoyl}piperidine-1-carboxylate
[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl](thiophen-2-yl)methanol
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[4-(morpholin-4-yl)butyl]amino}methyl)phenoxy]propan-2-ol