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N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-4-sulfamoylbenzamide
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1,2,5-thiadiazole-3-carboxamide
N-({8-[(2,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
5-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-[(2-hydroxyethyl)(propyl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
(2S,3R)-2-amino-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-hydroxybutan-1-one
(2E)-N-cyclopentyl-3-(1-methyl-1H-pyrazol-4-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)prop-2-enamide
2-cyclobutaneamido-7-oxo-N-(propan-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(3S)-1-[2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidin-3-ol
2-({4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
methyl (2S,4R)-1-[(4-ethylphenyl)methyl]-4-(4-fluorobenzamido)pyrrolidine-2-carboxylate
ethyl 1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxylate
7-(3,6-dimethylpyrazin-2-yl)-4-(pent-2-yn-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-amino-4-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-{[2-(2-phenylethynyl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
8-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-butyl-5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)amine
8-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-yl)-6-(1H-indole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
5-[1-(4-chlorophenyl)cyclopropyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(2R,3R)-2-methoxy-1'-(1-methylcyclohexanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
8-(pyrimidin-5-ylmethyl)-8-azaspiro[4.5]decane-7,9-dione
2-methoxyethyl N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
N-(2-methyl-1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
N-cyclopropyl-2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
4-acetamido-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
4-{[4-(trifluoromethoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1-[(6-chloropyridin-3-yl)methyl]-2-methyl-1,4-diazepan-5-one
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]urea
5-(azetidin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-ethyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(piperidin-1-yl)ethyl]piperidine-3-carboxamide
1-cyclobutyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-cyclopentyl-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
N-[(3-methoxy-2-propoxyphenyl)methyl]thiolan-3-amine
1-{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-methyl-1H-pyrrole-3-carboxamide
N-[2-(dimethylamino)-1-phenylethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-methyl-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
N-(9H-fluoren-9-yl)-6-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-[3-(dimethylamino)propyl]-8-[2-(ethylamino)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(1,2-oxazolidine-2-carbonyl)-2-(3-phenylpropyl)-1,3-benzoxazole
1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
2-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline
2-(2-ethylpiperidin-1-yl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one