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4-methyl-2-[1-(pyrrolidin-3-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
9-methoxy-N-methyl-3-[(5-methylthiophen-2-yl)methyl]-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4R)-1-(3-chloro-4-fluorobenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-2-{4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}acetamide
5-amino-4-chloro-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-ethyl-N-[(4-fluorophenyl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-(3-methoxypropyl)-3-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-3-phenylpyrrolidine-2,5-dione
methyl (2S,4S)-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]pyrrolidine-2-carboxylate
3-[(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
4-cyclobutaneamido-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-2,6-dimethylquinoline-4-carboxamide
4-chloro-2-fluoro-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)benzamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-2H-1,3-benzodioxole-5-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-cyclopentyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide
4-chloro-N,N-dimethyl-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
6-oxo-N-(2-phenylethyl)-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-{[3-methyl-7-(3-methylthiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
2-amino-6-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
1-{2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]phenyl}ethan-1-one
3-[3-({[2-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)-1H-indol-1-yl]propanamide
5-(3-methyl-3-phenylpiperidine-1-carbonyl)-2-(methylsulfanyl)pyrimidine
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}pent-4-en-1-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)benzonitrile
(3S,4S)-4-(pyrrolidin-1-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidin-3-ol
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
ethyl 5-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
11-{[(4-fluorophenyl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1,3-benzothiazol-2-yl)-4-(3-hydroxypropanoyl)-1,4-diazepane-6-carboxylic acid
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-[4-(hydroxymethyl)piperidine-1-carbonyl]-1-methylpyrrolidine-2-carboxylic acid
8-[(3,4-dimethylphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N,2-dimethyl-N-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4S)-3-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
methyl({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 4-[4-fluoro-3-(hydroxymethyl)phenyl]-2-(methylsulfanyl)pyrimidine-5-carboxylate
2-(3-fluorophenyl)-N-[(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
3-methyl-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
N-[2-(2,4-difluorophenyl)-1-{1-[3-(dimethylcarbamoyl)propanoyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
2-(dimethylamino)-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-cyclopentyl-5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]piperidin-2-one