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(2R)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylbutanamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(1-methylpiperidin-4-yl)benzamide
1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-4-phenylbutan-1-one
N-(2,4-dimethylphenyl)-3-[(3R)-3-hydroxypyrrolidin-1-yl]-3-oxopropanamide
5-(propan-2-yl)-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-oxo-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1,2-dihydroquinoline-4-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl](2-methylpropyl)amine
dimethyl({[4-methyl-5-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
N-(propan-2-yl)-3-propanamido-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
3-hydroxy-2-methyl-N-{[1-(2-phenylethyl)pyrrolidin-3-yl]methyl}benzamide
2-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]-1,2-oxazolidin-4-ol
2-(methylamino)-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
6-methoxy-2-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2,6,8-trimethylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
4-[7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(3-chlorophenoxy)ethan-1-one
3-(3-benzoylpiperidine-1-carbonyl)-4-phenyl-1H-pyrazol-5-amine
4-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-3-methylpiperazin-2-one
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-(2-aminoethyl)-N,5,6-trimethyl-N-(quinolin-8-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-methoxy-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
4-cyclopentyl-N-{[4-(dimethylamino)oxan-4-yl]methyl}pyrimidin-2-amine
1-[(3-chlorophenyl)methyl]-4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-[4-(dimethylamino)phenyl]propan-1-one
4-({1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-6-methyl-1,2-dihydropyridin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}thiophene-2-carboxamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
3-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanamide
(3aS,7aR)-5-methyl-2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-(ethylamino)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}pyrimidine-5-carboxamide
1-(1H-indazol-6-yl)-5-methyl-4-[2-(pyrazin-2-yl)acetyl]piperazin-2-one
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
3-{5-[(2E)-pent-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}propane-1,2-diol
1-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-(3-chloro-4-methoxyphenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
9-(cyclopropylmethyl)-4-[(3-fluoro-4-methylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl (2S,4S)-4-(5-hydroxypyrazine-2-amido)-1-methylpyrrolidine-2-carboxylate
4-(2,5-dichlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-ethyl-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
methyl 1-[(3S,5S)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
(3S,4R)-1-(4-carboxybutanoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,4-triazole-5-carboxamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
4-[(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-({4-[(dimethylamino)methyl]phenyl}methyl)-2-(3-methoxyphenyl)acetamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine