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(3R,5S)-N3-[2-(1H-imidazol-4-yl)ethyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-(thiolan-3-yl)pyrimidin-2-amine
1-(2-hydroxyethyl)-5,5-diphenylpiperidin-2-one
4-({2-[1-(oxane-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-chloro-N-({1-[2-(4-hydroxypiperidin-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
2-cyclopropyl-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-{4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-1-yl}phenol
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
N-(2-hydroxy-2-phenylethyl)-5-methanesulfonamido-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
8-[(4-fluoro-3-methoxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyridine-2-carbonitrile
1-[4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(2-chlorophenyl)methyl]-3-(2-ethyl-1H-imidazol-1-yl)-N-(prop-2-en-1-yl)propanamide
1-[(4-methylphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazin-2-one
(1S,5R)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(pyrrolidin-1-yl)acetamide
5-{4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
3-{[(5-chloropyridin-2-yl)amino]methyl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
(3S,4S)-4-[4-(benzyloxy)piperidin-1-yl]-1-(4-methoxybenzoyl)pyrrolidin-3-ol
3-(but-2-yn-1-yl)-5-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
1,3-dimethyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-5-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-cyclopropylpyrimidine
3-(azocan-1-yl)-N-[3-(morpholin-4-yl)propyl]propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-(pyrimidin-4-ylmethyl)-1,3-oxazole-4-carboxamide
4-benzyl-1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-ethyl-1,4-diazepan-5-one
2-({2-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
(5S,9aS,9bS)-5-[2-(cyclopentyloxy)phenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1λ6-thiomorpholine-1,1-dione
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
4-fluoro-N-{3-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-3-oxopropyl}benzamide
(3aR,6aR)-2-cyclopentyl-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
N-phenyl-1-[2-(pyridin-4-yl)quinoline-4-carbonyl]piperidin-3-amine
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(4-ethoxyphenyl)methyl]piperazin-2-one
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-4-(4-methylphenyl)piperazine
7-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one