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1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
(1S,5R)-N-[(3-fluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-benzyl-1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
5-(1-benzofuran-2-yl)-3-cyclopropyl-1H-1,2,4-triazole
N-(2-methyl-1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
1-{4-[(cyclopentylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[4-(3-methoxyphenyl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N,N,4-trimethyl-5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
1-(3-{[(quinolin-7-yl)carbamoyl]amino}propyl)piperidine-3-carboxamide
6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-[(2-chloro-5-fluorophenyl)methanesulfonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
3-[2-(4-methoxyphenyl)phenyl]-1-methyl-1-(oxan-2-ylmethyl)urea
4-methyl-6-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,3-benzothiazol-2-amine
N-methyl-5-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-({7-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
3-fluoro-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzene-1-sulfonamide
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
5-{3-[3-(2-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N-[(3S,4R)-1-(4-chlorobenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-({1-[1-(carbamoylmethyl)piperidine-3-carbonyl]azetidin-3-yl}oxy)benzoic acid
3-{1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]piperidin-3-yl}benzoic acid
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
[(3R,4R)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(2S)-2-amino-2-(2-chlorophenyl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-{[6-(4-methanesulfonylphenyl)quinazolin-4-yl]amino}ethan-1-ol
2-(2-methyl-1H-indol-3-yl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
3-{1-[(2,3-difluorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2,6-dihydroxy-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]benzamide
7-cyclopentyl-2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3-(3-methoxyphenyl)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(hydroxymethyl)cyclopentyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-({1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl)(4-methyl-1-phenylpentyl)amine
4-{[1-(hydroxymethyl)cyclobutyl]methyl}-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
N-[(5-methylfuran-2-yl)methyl]-3-[1-(2,2,2-trifluoroethanesulfonyl)piperidin-3-yl]propanamide
2-{4-[(2,3-difluorophenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4-fluorophenyl)propan-1-one