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3-{2-[4-(aminomethyl)piperidin-1-yl]-2-oxoethyl}-3-benzyl-1-methyl-2,3-dihydro-1H-indol-2-one
(2S,4S)-4-[4-({[(5-fluoro-2-methylphenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-methyl-3-(pyrrolidin-3-yl)-N-(quinolin-5-ylmethyl)benzamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-one
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
2-[2-(1H-imidazol-4-yl)ethyl]-8-[5-(methoxymethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-methoxy-N-[3-(2-{[methyl(propan-2-yl)amino]methyl}propanamido)phenyl]benzamide
N-(6-phenoxypyridin-3-yl)-1-(thiophene-2-carbonyl)piperidine-4-carboxamide
1-benzyl-4-oxo-N-(prop-2-en-1-yl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-[(oxolan-3-yl)amino]pyridine-3-carboxamide
2-(1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-5-methyl-1H-1,3-benzodiazole
3-{[1-(3-methoxy-2,2-dimethylpropanoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-5,6,7,8-tetrahydroquinazolin-2-amine
6-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-phenoxyacetamide
2-{1-[(4-fluorophenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
5-(1-cyclohexanecarbonylpiperidin-4-yl)-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
1-(diphenylmethyl)-N-(1-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-(4-methoxy-2-methylphenyl)-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-{[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(piperidin-1-yl)ethan-1-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
(4aR,7aS)-1-acetyl-4-(5-methyl-1H-indole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
[(3R,4S)-1-benzyl-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-3-(naphthalen-1-ylmethyl)-N-(1,3-thiazol-4-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(cyclohexylmethyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-3-phenylpyrrolidine-2,5-dione
methyl 6-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[1-(pyridin-4-yl)propyl]propanamide
3-(2-fluorophenyl)-6-(2-methyl-1,3-thiazole-4-carbonyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
3-ethyl-N-({7-[2-(2-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
1-benzyl-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(5-acetylthiophen-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-{[1-(2-phenylethyl)piperidin-4-yl]methyl}urea
3-methyl-1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}butan-1-one
N-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}acetamide
(2E)-3-(2-fluorophenyl)-N-{[3-methyl-7-(5-methylpyrazine-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}prop-2-enamide
8-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(5-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-propyl-1H-pyrazole-5-carboxamide
1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-{ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid