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ethyl 4-{2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
7-methyl-4-{2-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-methyl-1-(4-{5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
3-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
3-fluoro-N-[(8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
3-methyl-4-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
5-[2-(benzylamino)ethyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]pyrrolidin-2-one
3-[3-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-indol-1-yl]propanamide
5-[(3S)-3-ethylmorpholine-4-carbonyl]-2-methyl-1,3-benzothiazole
4-methyl-2-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
propyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
N-phenyl-5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]methanol
N-(1-benzylpiperidin-3-yl)-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1'-(4-methyl-1H-imidazole-5-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-(2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}ethan-1-one
1-{[4-(benzyloxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
(1R,5R)-6-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-(4-methylpiperazin-1-yl)propanamide
2-(3-fluorophenyl)-8-methoxy-5-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-{[(3S)-3-aminopyrrolidin-1-yl]sulfonyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-[(2R,3R)-1'-(2H-1,3-benzodioxole-5-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
4-ethyl-3-[1-(4-hydroxybenzoyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-3,9-diazaspiro[5.5]undecane
methyl 5-cyano-2-methyl-6-[4-(morpholin-4-ylmethyl)piperidin-1-yl]pyridine-3-carboxylate
3-[(3R,4S)-4-(dimethylamino)-1-(2-hydroxy-4-methylbenzoyl)piperidin-3-yl]propanoic acid
5-[(3R,4S)-3-(2-carboxyethyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]thiophene-2-carboxylic acid
4-{3-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
5-benzenesulfonamido-1-ethyl-N,2-dimethyl-N-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(2-phenylpropanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)carbamoyl]methyl}piperidine-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 2-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}-1,3-oxazole-4-carboxylate
benzyl(cyclopropylmethyl){[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
3-tert-butyl-1-methyl-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(4-fluorophenyl)-N-methyl-4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
2-(dimethylamino)-7-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{2-[(4-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(pyridin-3-yl)propyl]piperidin-4-amine
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-[2-oxo-2-(3-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
(1R,5R)-6-[(1-ethyl-1H-indol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane