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N-(1,3-dihydro-2-benzofuran-5-yl)-2-(pyrrolidin-3-yl)benzamide
1-benzyl-4-[3-(diphenylmethyl)-1,2-oxazole-5-carbonyl]piperazine
2-(azepan-1-yl)-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-({4-[4-(1H-imidazol-1-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenol
1-[(4aR,8aR)-4a-hydroxy-7-[(4-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(phenylamino)pyrimidine-5-carboxamide
2-methoxy-5-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
1-methyl-4-({4-methyl-5-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1-methylcyclopropanecarbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5,7-dimethyl-N-[2-(morpholin-4-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-(4-{5-methyl-4-[(3-methylbutanamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
5-chloro-2-methoxy-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
(5S,9aS,9bS)-2-cyclopentyl-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{[4-(4-hydroxy-2-methylquinolin-8-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
3,3-dimethyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}butanamide
4,6-dimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}-6-methyl-4H-chromen-4-one
(benzylsulfamoyl)({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
7-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decane
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-[3-(pyridin-3-yl)propyl]urea
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-phenyl-1H-pyrazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-5-(oxan-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-(pyridin-3-yl)-N-[1-(thian-4-yl)piperidin-4-yl]pyrimidin-2-amine
N-[(3,4-dimethoxyphenyl)methyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-(2-phenylquinoline-4-carbonyl)pyrrolidine-2-carboxamide
1-(piperidine-1-sulfonyl)-4-(pyrimidin-4-yl)-1,4-diazepane
6-{[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,7aS)-1-methyl-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
3-[(3,5-difluorophenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(5S,9aS,9bS)-5-(1-phenyl-1H-pyrazol-4-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-cyclopentyl-2-[4-(1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-(4-propylmorpholin-3-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}acetamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[(4-fluorophenyl)methyl]piperidine
6-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile
6-methyl-2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
(2R)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidine-2-carboxamide
8-[(3,4-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[(2R,5S)-5-[(3-fluoro-4-methoxyphenyl)methyl]oxolan-2-yl]methyl}-1,4-oxazepane