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N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-ol
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3,5-dimethyl-1H-indole-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(2-ethylpyrimidine-5-carbonyl)-4-methanesulfonyl-1,4-diazepane
3-ethyl-2-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1H-indole
1-(cyclohex-3-ene-1-carbonyl)-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-cyclopentyl-N'-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}ethanediamide
ethyl 5-(1H-1,3-benzodiazole-5-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(3-methylpyridin-2-yl)-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazine
2-phenyl-1-{4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
2-{2-[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridine
N-(2,3-dimethylphenyl)-2-{[4-(furan-2-yl)butan-2-yl]amino}acetamide
1-[2-(3-methoxyphenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
(2-{[4-(2-amino-4-methylpyrimidine-5-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
N-(2,2-dimethyloxan-4-yl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-acetyl-8-(benzylcarbamoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,1-dimethyl-3-(2-methylpropyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
1-(1-ethylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(2-methyl-1-benzofuran-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-(1-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
1-(2-methylphenyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-N-methylpyridin-2-amine
2-{3-cyclopentyl-5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-cyclohexyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-(1-cyclopropanecarbonylpiperidin-3-yl)-4-pentanamidobenzamide
1-ethyl-3-(3-fluoro-4-methylphenyl)-6-[(2-methyl-1,3-thiazol-5-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[methyl(piperidin-4-yl)amino]-N-{[4-(trifluoromethoxy)phenyl]methyl}acetamide
4-[1-(4-methoxyphenyl)-2,2-dimethylcyclopropanecarbonyl]thiomorpholine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methoxy-3-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-indol-1-yl)propyl]acetamide
8-(2H-1,3-benzodioxole-5-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
6-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-N,N,1-trimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
1-(furan-3-ylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-{1-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-2-methyl-1-oxopropan-2-yl}acetamide
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pyridine-3-carboxylic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyrimidin-2-ylsulfanyl)acetamide
7-(2-oxo-1,3-oxazolidin-3-yl)-4-(1-phenyl-1H-pyrazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-5-(3-phenylpiperidine-1-carbonyl)pyrimidin-4-ol
2-{2-oxo-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
4-[7-(6-methylpyridine-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
methyl 1-[(3R,5S)-5-(cycloheptylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate