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2-(3-chloro-5-fluorophenyl)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
(3R,4R)-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(hydroxymethyl)piperidin-3-ol
1-(1-benzothiophen-2-ylmethyl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(4-methoxyphenyl)-2-methylpiperazine
2-acetyl-8-(naphthalen-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
N-(cyclopent-3-en-1-yl)-2-{4-[3-(3-methoxyphenyl)propanoyl]morpholin-3-yl}acetamide
4-benzoyl-1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
N-[2-(2,4-difluorophenyl)-1-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
methyl 1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-2-carboxylate
4-(3,6-dimethylpyrazin-2-yl)-2-{[methyl(2-phenylethyl)amino]methyl}phenol
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(thiophen-2-yl)ethyl]propanamide
1-cyclobutanecarbonyl-4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
5-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
4-[1-(2-phenoxyethyl)-1H-imidazol-2-yl]benzonitrile
methyl 6-[(2-hydroxyphenyl)methyl]-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(1H-imidazol-1-yl)propanamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
(3S,4R)-1-(6-aminopyrimidin-4-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
1-[(4-methanesulfonylphenyl)methyl]-2-(1,3-thiazol-2-yl)piperidine
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]propan-1-one
2-cyano-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylbenzamide
5-{2-[(prop-2-en-1-yl)amino]ethyl}-1-[3-(pyridin-4-yl)propyl]pyrrolidin-2-one
[(3-methyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
N-[2-(3-methoxyphenyl)phenyl]-1-(quinolin-5-ylmethyl)piperidine-4-carboxamide
5-(2-fluorophenyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(1-ethylcyclopropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(naphthalene-1-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
N-(2-hydroxyethyl)-N-(2-methylpropyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2,3-dimethoxy-N-methylbenzamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-methyl-7-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N,N,4-trimethyl-3-{[(2-propoxyethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
3-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one