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N-[1-(1-benzoylpiperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N-methylcyclopropanecarboxamide
2-(2,5-dimethylphenyl)-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}ethan-1-one
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-pyrazole-4-carboxamide
N-(1-methyl-1H-pyrazol-4-yl)-2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]acetamide
(3aS,6aR)-5-(4-amino-5-methylpyrimidin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(3-fluorophenyl)-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-(1H-imidazol-2-ylmethyl)-1-(2-methylpropyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-cyclohexyl-1-cyclopropyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
1-cyclopentyl-4-(1H-imidazol-4-ylmethyl)piperazin-2-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]benzamide
4-{1-benzyl-5-[(2S,4R)-4-hydroxypyrrolidin-2-yl]-1H-1,2,4-triazol-3-yl}benzamide
N-cyclopropyl-2,4-difluoro-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)benzene-1-sulfonamide
N-cyclopropyl-4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4,6-dimethylpyridine-3-carboxamide
1'-(5-ethyl-1,3,4-oxadiazol-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
3-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
1-(3-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-[(2R,3R)-2-ethoxy-1'-[(5-methylfuran-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclobutanecarboxamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
(2E)-3-(2-chlorophenyl)-N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}prop-2-enamide
3-butyl-4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-methylpiperazin-2-one
(2S)-2-amino-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
6-cyclopropyl-N-[(3R,4S)-4-cyclopropyl-1-(oxane-4-carbonyl)pyrrolidin-3-yl]pyrimidin-4-amine
6-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-({[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
2-methoxy-5-[(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
6-fluoro-2-{[4-(3-hydroxyphenyl)piperazin-1-yl]methyl}quinolin-4-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-methanesulfonamidoacetamide
3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
1-(azepan-1-yl)-2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-methyl-4-(4-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}phenyl)butan-2-ol
N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(5-propylfuran-2-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
(2R,3R)-1'-(pyrimidin-2-yl)-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl})amine
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidine
4-{[(1R,5S,6R)-3-(3-cyclohexylpropanoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}-1λ6-thiomorpholine-1,1-dione
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(pyridin-2-yl)acetamido]pyrrolidine-2-carboxamide
4-{[1-(2-methoxypyridine-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
5-{[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
5-(4-acetylphenoxymethyl)-N-methyl-N-(4-methylpentan-2-yl)-1,2-oxazole-3-carboxamide