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4-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
2-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
3-{[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}-5-methyl-1,2,4-oxadiazole
N-{[7-(4-tert-butylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(2R)-2-cyclohexyl-2-hydroxy-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-cyclopentyl-2-methoxy-3-{[(6-methoxypyrimidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carboxamide
(4S)-4-acetamido-5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-oxopentanamide
3-(3,4-dimethoxybenzoyl)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
1-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}imidazolidin-2-one
2-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
7-(cyclopropylmethyl)-2-methyl-N-[2-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-(2-fluorophenyl)-N-methyl-N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}-5-(propan-2-yl)-1,2-oxazole
1-[1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}furan-2-carboxamide
1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-(furan-3-carbonyl)-1,4-diazepane
N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
4-(1H-pyrazol-3-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}benzamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-acetyl-N-(1-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
3-ethyl-8-[3-(methylsulfanyl)butyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1,4-dithiepan-6-amine
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S,5S)-1-benzyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}pyrrolidin-3-amine
1-tert-butyl-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
N-({3-methyl-7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-indole-2-carboxamide
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-(2-ethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{methyl[(4-methyl-5-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
2-(3-phenylpropyl)-8-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
(1R,2R)-2-[propyl({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl})amino]cyclohexan-1-ol
2-(2-chlorophenyl)-2-hydroxy-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
4-benzyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-one
(2R)-2-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}propanamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-4-carboxamide
N-cyclopropyl-6-[4-(1-ethoxyethyl)phenyl]pyridazin-3-amine
3-[5-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenol
1-(2-methoxyphenyl)-2,2-dimethyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-N-[(2-methoxyphenyl)methyl]acetamide
N-(furan-2-ylmethyl)-N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-[3-({[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
3-[(2-acetamidoethyl)sulfamoyl]-N-(oxan-3-ylmethyl)benzamide
(4aS,8aS)-2-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-decahydroisoquinolin-4a-ol
N-{[7-(3-fluoro-4-methoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide