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N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(furan-2-ylmethyl)-2-[5-oxo-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
3-[5-(1-methyl-1H-indole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(3S,4R)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-(3-methyl-1-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-3-carboxamide
N-(2,5-dimethylphenyl)-3-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
N4,N4,N6-trimethyl-N6-[(3-methylpyridin-4-yl)methyl]pyrimidine-4,6-diamine
(cyclopropylmethyl)(oxolan-2-ylmethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidine
1-(2-aminoethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-ethyl-4-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperazin-2-one
2-(dimethylamino)-2-(4-methylphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
2-[(4-phenylazepan-1-yl)methyl]pyridine-3-carboxylic acid
1-(5-ethylpyrimidin-2-yl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]morpholine-2-carboxamide
2-{2-[(thiolan-3-yl)amino]ethyl}-3,4-dihydroquinazolin-4-one
N-[(5-methylfuran-2-yl)methyl]-3-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-3-yl}propanamide
N-[2-(cyclohex-3-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-[(4-aminopiperidin-1-yl)sulfonyl]-N-[2-(1H-pyrrol-1-yl)ethyl]benzamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
N-(pyridin-4-ylmethyl)-4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2,4,6-trifluorophenyl)ethan-1-one
5-(morpholin-4-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(diethylamino)ethyl]-N-methylbenzamide
1-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methylbenzamide
3-methyl-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[2-(pyridin-3-yloxy)phenyl]urea
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(2-methoxyphenyl)methyl]piperidine-4-carboxamide
2-methyl-N-[2-(quinolin-8-yloxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4aR,7aS)-1-benzoyl-4-(1-methylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)phenol
1-methyl-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-1-(quinolin-3-ylmethyl)urea
(2S,4S)-4-amino-1-(2-cyclopropylquinoline-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-benzyl-3-({[(4-ethylphenyl)methyl](methyl)amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-ethyl-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-3-methylpiperidine-3-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
1-[7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
(3R,4R)-4-cyclopropyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-methylpiperidin-4-ol
{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
2-{3-[2-(4-fluorophenoxy)ethyl]phenoxy}propanamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-benzyl-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(2R,3R)-1'-[(4-acetamidophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-(aminomethyl)-4-(2-methoxy-5-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one